Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50028904
TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM22971(Meclofenamate | CHEMBL509 | 2-[(2,6-dichloro-3-met...)
Affinity DataIC50: 100nMAssay Description:Compound was evaluated in an intact RBL-1 cell line for inhibition of 5-CyclooxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280051(5-[2-(3-Trifluoromethyl-phenylamino)-pyridin-3-yl]...)
Affinity DataIC50: 190nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048004(5-(2-(3-(trifluoromethyl)phenylamino)phenyl)-1,3,4...)
Affinity DataIC50: 270nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048003(5-[2-(2,3-Dimethyl-phenylamino)-phenyl]-[1,3,4]oxa...)
Affinity DataIC50: 610nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048007(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-3...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50048007(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-3...)
Affinity DataIC50: 740nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50048004(5-(2-(3-(trifluoromethyl)phenylamino)phenyl)-1,3,4...)
Affinity DataIC50: 770nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50047998(5-[2-(3-Trifluoromethyl-phenylamino)-phenyl]-3H-[1...)
Affinity DataIC50: 850nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50047998(5-[2-(3-Trifluoromethyl-phenylamino)-phenyl]-3H-[1...)
Affinity DataIC50: 870nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280051(5-[2-(3-Trifluoromethyl-phenylamino)-pyridin-3-yl]...)
Affinity DataIC50: 990nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50048003(5-[2-(2,3-Dimethyl-phenylamino)-phenyl]-[1,3,4]oxa...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50048009(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-[...)
Affinity DataIC50: 1.39E+3nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048009(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-[...)
Affinity DataIC50: 1.75E+3nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM22971(Meclofenamate | CHEMBL509 | 2-[(2,6-dichloro-3-met...)
Affinity DataIC50: 2.40E+4nMAssay Description:Compound was evaluated in an intact RBL-1 cell line for inhibition of 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article