Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50021845
Displayed 1 to 50 (of 61 total ) | Next | Last >>
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human P2X3 receptor expressed in 1321N1 cells assessed as reduction in calcium level preincubated for 30 mins followed by alph...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321N1 cells assessed as reduction in calcium level preincubated for 3 mins followed by alp...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human P2X3 receptor assessed as reduction in calcium level incubated for 18 hrs by Fluo-4 AM dye based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Antagonist activity at human P2X3 receptor expressed in 1321N1 cells assessed as reduction in calcium level preincubated for 3 mins followed by alpha...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human P2X3 receptor expressed in HEK293 cells preincubated for 30 mins followed by alpha, beta me-ATP addition and measured fo...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human P2X3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human P2X3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Antagonist activity at human P2X2/3 receptor assessed as reduction in calcium level incubated for 18 hrs by Fluo-4 AM dye based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 133nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 162nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 163nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321N1 cells assessed as reduction in calcium level preincubated for 30 mins followed by al...More data for this Ligand-Target Pair
Affinity DataIC50: 288nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 301nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 362nMAssay Description:Antagonist activity at alpha, beta-meATP activated human P2X3 receptor by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Antagonist activity at human P2X2/3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 542nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 547nMAssay Description:Antagonist activity at rat P2X2/3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 602nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 659nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 722nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 763nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 764nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 798nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 811nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 881nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 994nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 995nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 995nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.19E+3nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+3nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+3nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.45E+3nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+3nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.03E+3nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Antagonist activity at human P2X2/3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.28E+3nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair






3D Structure (crystal)


























