Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50021891
TargetCyclin-dependent protein kinase PHO85(Baker's yeast)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataEC50:  31nMAssay Description:Binding affinity to yeast Pho85 pretreated with yeast lysates for 45 mins followed by incubation with Kinobead-Sepharose affinity matrix slurry for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645820(CHEMBL5592073)
Affinity DataEC50:  130nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataEC50:  140nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645822(CHEMBL5579744)
Affinity DataEC50:  230nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataEC50:  300nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645815(CHEMBL5590260)
Affinity DataEC50:  330nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645820(CHEMBL5592073)
Affinity DataEC50:  350nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645820(CHEMBL5592073)
Affinity DataEC50:  570nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataEC50:  610nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataIC50: 640nMAssay Description:Inhibition of CDK2 in human OVCAR-3 cells assessed as reduction in Rb phosphorylation at T821 residue treated for 4 hrs followed by drug wash-out and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645823(CHEMBL5595750)
Affinity DataEC50:  700nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645819(CHEMBL5591069)
Affinity DataEC50:  870nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645814(CHEMBL5590401)
Affinity DataEC50:  900nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataIC50: 950nMAssay Description:Inhibition of CDK2 in human OVCAR-3 cells assessed as reduction in Rb phosphorylation at T821 residue treated for 4 hrs followed by drug wash-out and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645821(CHEMBL5591436)
Affinity DataEC50:  990nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK2 in human OVCAR-3 cells assessed as reduction in Rb phosphorylation at T821 residue measured after 120 hrs by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645822(CHEMBL5579744)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of CDK2 in human OVCAR-3 cells assessed as reduction in Rb phosphorylation at T821 residue measured after 18 hrs by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645827(CHEMBL5595307)
Affinity DataEC50:  1.40E+3nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645825(CHEMBL5591862)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645815(CHEMBL5590260)
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645825(CHEMBL5591862)
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645818(CHEMBL5592346)
Affinity DataEC50:  1.62E+3nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645827(CHEMBL5595307)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645810(CHEMBL5589612)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human full length CDK2 (1 to 298 residues)/N-terminal GST-tagged Cyclin E1 (1 to 410 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645814(CHEMBL5590401)
Affinity DataEC50:  2.89E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645816(CHEMBL5583972)
Affinity DataEC50:  3.00E+3nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645813(CHEMBL5595148)
Affinity DataIC50: 3.00E+3nMAssay Description:Reversible inhibition of human full length CDK2 (1 to 298 residues)/N-terminal GST-tagged Cyclin E1 (1 to 410 residues) expressed in baculovirus expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645822(CHEMBL5579744)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645815(CHEMBL5590260)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645825(CHEMBL5591862)
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645823(CHEMBL5595750)
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645821(CHEMBL5591436)
Affinity DataEC50:  5.25E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645814(CHEMBL5590401)
Affinity DataEC50:  5.36E+3nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645821(CHEMBL5591436)
Affinity DataEC50:  5.76E+3nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645826(CHEMBL5593130)
Affinity DataEC50:  6.10E+3nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645826(CHEMBL5593130)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645827(CHEMBL5595307)
Affinity DataEC50:  6.50E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645813(CHEMBL5595148)
Affinity DataIC50: 7.00E+3nMAssay Description:Reversible inhibition of human full length CDK1 (1 to 297 residues)/N-terminal GST-fused Cyclin B1 (1 to 433 residues) expressed in baculovirus expre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645816(CHEMBL5583972)
Affinity DataEC50:  8.00E+3nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645812(CHEMBL5590952)
Affinity DataIC50: 9.00E+3nMAssay Description:Reversible inhibition of human full length CDK2 (1 to 298 residues)/N-terminal GST-tagged Cyclin E1 (1 to 410 residues) expressed in baculovirus expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645813(CHEMBL5595148)
Affinity DataIC50: 9.00E+3nMAssay Description:Reversible inhibition of human full length CDK7 (1 to 346 residues)/N-terminal GST-fused Cyclin H (1 to 323 residues)/MAT1 (1 to 309 residues) expres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645816(CHEMBL5583972)
Affinity DataEC50:  1.16E+4nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645823(CHEMBL5595750)
Affinity DataEC50:  1.22E+4nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645818(CHEMBL5592346)
Affinity DataEC50:  1.64E+4nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645826(CHEMBL5593130)
Affinity DataEC50:  1.77E+4nMAssay Description:Inhibition of CDK1/Cyclin B1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645812(CHEMBL5590952)
Affinity DataIC50: 1.90E+4nMAssay Description:Reversible inhibition of human full length CDK1 (1 to 297 residues)/N-terminal GST-fused Cyclin B1 (1 to 433 residues) expressed in baculovirus expre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645812(CHEMBL5590952)
Affinity DataEC50:  2.20E+4nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645817(CHEMBL5594039)
Affinity DataEC50:  2.66E+4nMAssay Description:Inhibition of CDK2/Cyclin E1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
LifeMine Therapeutics

Curated by ChEMBL
LigandPNGBDBM50645818(CHEMBL5592346)
Affinity DataEC50:  3.02E+4nMAssay Description:Inhibition of CDK7/Cyclin H/MAT1 NanoLuc fusion vector (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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