Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50021382
Affinity DataIC50: 7.60nMAssay Description:Inhibition of GST-tagged LC3B (unknown origin) using biotin-labeled LBP2 as substrate preincubated with compound for 12 hrs followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of GST-tagged wild type LC3B (unknown origin) using biotin-labeled LBP2 as substrate preincubated with compound for 12 hrs followed by sub...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of LC3B (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of LC3A (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of GST-tagged LC3B (unknown origin) using biotin-labeled LBP2 as substrate preincubated with compound for 12 hrs followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of GST-tagged LC3B (unknown origin) using biotin-labeled LBP2 as substrate preincubated with compound for 12 hrs followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of GST-tagged LC3B K49R mutant (unknown origin) using biotin-labeled LBP2 as substrate preincubated with compound for 12 hrs followed by s...More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor-associated protein-like 2(Homo sapiens)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Inhibition of GABARAPL2 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 920nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 950nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor-associated protein-like 1(Homo sapiens)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of GABARAPL1 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.44E+3nMAssay Description:Inhibition of GABARAP (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
TargetMicrotubule-associated protein 1 light chain 3 gamma(Homo sapiens)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataIC50: 4.52E+3nMAssay Description:Inhibition of LC3C (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.77E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.14E+3nMAssay Description:Inhibition of N-terminal GST-tagged LC3B (unknown origin) measured for 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.07E+3nMAssay Description:Binding affinity to N-terminal GST-tagged LC3B (unknown origin) assessed as inhibition constant measured for 18 hrs by fluorescence polarization assa...More data for this Ligand-Target Pair
Affinity DataKi: 7.22E+4nMAssay Description:Binding affinity to N-terminal GST-tagged LC3B (unknown origin) assessed as inhibition constant measured for 18 hrs by fluorescence polarization assa...More data for this Ligand-Target Pair
Affinity DataKi: 8.63E+4nMAssay Description:Binding affinity to N-terminal GST-tagged LC3B (unknown origin) assessed as inhibition constant measured for 18 hrs by fluorescence polarization assa...More data for this Ligand-Target Pair





























