Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50020935
Displayed 1 to 50 (of 62 total ) | Next | Last >>
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of BRD4 BD1/2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 103nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inhibition of BRD4 BD1/2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Inhibition of BRD3 BD1/2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 127nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 153nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 165nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 199nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 264nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 268nMAssay Description:Inhibition of BRD3 BD1/2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 276nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 309nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 315nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 319nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 319nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 354nMAssay Description:Inhibition of BRDT BD1 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 387nMAssay Description:Inhibition of BRD4 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 401nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 433nMAssay Description:Inhibition of BRDT BD1 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 456nMAssay Description:Inhibition of recombinant NAMPT (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 489nMAssay Description:Inhibition of BRD2 BD1/2 (unknown origin) incubated for 120 mins by TR-FRET assayMore data for this Ligand-Target Pair





3D Structure (crystal)



















