Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50022106
Affinity DataKd: 600nMAssay Description:Binding affinity to KLHL20 (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 670nMAssay Description:Binding affinity to human N-terminal KLHL3 (290 to 587 residues) extracted from Escherichia coli BL21 (DE3) assessed as dissociation constant by fluo...More data for this Ligand-Target Pair
Affinity DataKd: 690nMAssay Description:Binding affinity to KLHL3 (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+4nMAssay Description:Binding affinity to KLHL12 (unknown origin) extracted from Escherichia coli BL21 Gold (DE3) assessed as dissociation constant by fluorescence polariz...More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+4nMAssay Description:Binding affinity to KLHL12 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3.44E+4nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair




