Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50022106
TargetKelch-like protein 20(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50648228(CHEMBL5613204)
Affinity DataKd:  600nMAssay Description:Binding affinity to KLHL20 (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetKelch-like protein 3(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50648225(CHEMBL5611958)
Affinity DataKd:  670nMAssay Description:Binding affinity to human N-terminal KLHL3 (290 to 587 residues) extracted from Escherichia coli BL21 (DE3) assessed as dissociation constant by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetKelch-like protein 3(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50648224(CHEMBL5613311)
Affinity DataKd:  690nMAssay Description:Binding affinity to KLHL3 (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetKelch-like protein 12(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50648226(CHEMBL5612301)
Affinity DataKd:  1.50E+4nMAssay Description:Binding affinity to KLHL12 (unknown origin) extracted from Escherichia coli BL21 Gold (DE3) assessed as dissociation constant by fluorescence polariz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetKelch-like protein 12(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50648226(CHEMBL5612301)
Affinity DataKi:  2.10E+4nMAssay Description:Binding affinity to KLHL12 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50648227(CHEMBL5614112)
Affinity DataIC50: 3.44E+4nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed