Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50020785
TargetTyrosine-protein kinase JAK3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50633569(CHEMBL5421894)
Affinity DataIC50: 520nMAssay Description:Inhibition of N-terminal His-tagged human JAK3 (795 to 1124 residues) expressed in Sf21 cells incubated for 30 mins in presence of ATP by LANCE Ultra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50633569(CHEMBL5421894)
Affinity DataIC50: 530nMAssay Description:Inhibition of N-terminal GST-tagged human TYK2 (871to 1187 residues) expressed in Sf21 cells incubated for 30 mins in presence of ATP by LANCE Ultra ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50633569(CHEMBL5421894)
Affinity DataIC50: 840nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 (850 to 1154 residues) expressed in Sf21 cells incubated for 30 mins in presence of ATP by LANCE Ultra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50633569(CHEMBL5421894)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of N-terminal His-tagged human JAK2 (826 to 1132 residues) expressed in Sf21 cells incubated for 30 mins in presence of ATP by LANCE Ultra...More data for this Ligand-Target Pair
In DepthDetails
PubMed