Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50020783
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633561(CHEMBL5404503)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633562(CHEMBL5410813)
Affinity DataEC50:  8.50E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633563(CHEMBL5421918)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633564(CHEMBL5433171)
Affinity DataEC50:  6.90E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633565(CHEMBL5437877)
Affinity DataEC50:  1.03E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633566(CHEMBL5404545)
Affinity DataEC50:  2.83E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633567(CHEMBL5424611)
Affinity DataEC50:  8.80E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633568(CHEMBL5432734)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50541574(CHEMBL4636830)
Affinity DataEC50:  7.80E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50532217(CHEBI:67081 | Cannabigerolic Acid)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50318487(Cannabigerol | CHEMBL497318)
Affinity DataEC50:  700nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633560(CHEMBL5415604)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50318487(Cannabigerol | CHEMBL497318)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633563(CHEMBL5421918)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50532217(CHEBI:67081 | Cannabigerolic Acid)
Affinity DataIC50: 1.31E+3nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50541574(CHEMBL4636830)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633564(CHEMBL5433171)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633562(CHEMBL5410813)
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50532217(CHEBI:67081 | Cannabigerolic Acid)
Affinity DataIC50: 7.14E+3nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633563(CHEMBL5421918)
Affinity DataIC50: 7.90E+3nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633567(CHEMBL5424611)
Affinity DataIC50: 8.00E+3nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50541574(CHEMBL4636830)
Affinity DataIC50: 8.40E+3nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633560(CHEMBL5415604)
Affinity DataIC50: 1.04E+4nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50318487(Cannabigerol | CHEMBL497318)
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633564(CHEMBL5433171)
Affinity DataIC50: 1.39E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633565(CHEMBL5437877)
Affinity DataIC50: 1.73E+4nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633568(CHEMBL5432734)
Affinity DataIC50: 1.79E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633567(CHEMBL5424611)
Affinity DataIC50: 1.92E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633568(CHEMBL5432734)
Affinity DataIC50: 2.39E+4nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633565(CHEMBL5437877)
Affinity DataIC50: 2.51E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633566(CHEMBL5404545)
Affinity DataIC50: 2.95E+4nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633561(CHEMBL5404503)
Affinity DataIC50: 3.30E+4nMAssay Description:Antagonist activity at rat TRPM8 transfected in HEK293 cells assessed as inhibition of icilin induced increase in intracellular Ca2+ concentration pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633560(CHEMBL5415604)
Affinity DataIC50: 3.73E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633566(CHEMBL5404545)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633562(CHEMBL5410813)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50633561(CHEMBL5404503)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPA1 transfected in HEK293 cells assessed as desensitization by measuring inhibition of AITC induced increase in intracel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed