Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50019618
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50366237(GAMBOGIC ACID)
Affinity DataIC50: 176nMAssay Description:Inhibition of recombinant Bfl-1 (1-152) (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50610577(CHEMBL5283368)
Affinity DataIC50: 800nMAssay Description:Inhibition of Bfl-1 (unknown origin) incubated for 30 min by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50604878(CHEMBL5206188)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant Bfl-1 (unknown origin) expressed in Escherichia coli LOBSTR BL21 incubated for 1 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50610577(CHEMBL5283368)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of GST-tagged Bfl-1 (unknown origin) incubated for 60 min by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM34188(SMR000082310 | cid_2980973 | ethyl 2-[4-(4-fluorop...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of GST-tagged Bfl-1 (unknown origin) incubated for 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM34188(SMR000082310 | cid_2980973 | ethyl 2-[4-(4-fluorop...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) incubated in dark by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50013839(CHEMBL2030270)
Affinity DataIC50: 4.61E+3nMAssay Description:Inhibition of recombinant Bfl-1 (1-152) (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM53290(2-[4-[(4-bromophenyl)sulfonylamino]-1-hydroxynapht...)
Affinity DataIC50: 8.41E+3nMAssay Description:Inhibition of recombinant Bfl-1 (1-152) (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-like protein 1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM34188(SMR000082310 | cid_2980973 | ethyl 2-[4-(4-fluorop...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST fused Bcl-xL (unknown origin) incubated for 5 min by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetApoptosis regulator Bcl-2(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM34188(SMR000082310 | cid_2980973 | ethyl 2-[4-(4-fluorop...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST fused Bcl-2 (unknown origin) incubated for 5 min by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-like protein 2(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM34188(SMR000082310 | cid_2980973 | ethyl 2-[4-(4-fluorop...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST fused Bcl-w (unknown origin) incubated for 5 min by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM34188(SMR000082310 | cid_2980973 | ethyl 2-[4-(4-fluorop...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST fused Mcl-1 (unknown origin) incubated for 5 min by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621106(CHEMBL5401950)
Affinity DataKi:  630nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621105(CHEMBL5420281)
Affinity DataKi:  750nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50013888(CHEMBL3260038)
Affinity DataKi:  1.09E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621104(CHEMBL5440532)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621102(CHEMBL5438295)
Affinity DataKi:  1.63E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621099(CHEMBL5413651)
Affinity DataKi:  1.84E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM53290(2-[4-[(4-bromophenyl)sulfonylamino]-1-hydroxynapht...)
Affinity DataKi:  1.91E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621100(CHEMBL5418778)
Affinity DataKi:  1.92E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621098(CHEMBL5433077)
Affinity DataKi:  1.97E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50013862(CHEMBL3265294)
Affinity DataKi:  2.21E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50013834(CHEMBL3260039)
Affinity DataKi:  3.01E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM53290(2-[4-[(4-bromophenyl)sulfonylamino]-1-hydroxynapht...)
Affinity DataKi:  3.17E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50013885(CHEMBL3260035)
Affinity DataKi:  3.23E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50013862(CHEMBL3265294)
Affinity DataKi:  4.71E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50621105(CHEMBL5420281)
Affinity DataKi:  4.79E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50013888(CHEMBL3260038)
Affinity DataKi:  4.89E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50621104(CHEMBL5440532)
Affinity DataKi:  5.91E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621101(CHEMBL5438598)
Affinity DataKi:  6.19E+3nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50621102(CHEMBL5438295)
Affinity DataKi:  6.61E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50621106(CHEMBL5401950)
Affinity DataKi:  6.77E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50621100(CHEMBL5418778)
Affinity DataKi:  7.48E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
LigandPNGBDBM50013885(CHEMBL3260035)
Affinity DataKi:  8.64E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621096(CHEMBL5421542)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621097(CHEMBL5394425)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50621103(CHEMBL5415310)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of Bfl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed