Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50020088
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626067(CHEMBL5403042)
Affinity DataIC50: 0.160nMAssay Description:Displacement of [35S]MK-0677 from human GHSR1a expressed in HEK293 cell membrane by filter binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626066(CHEMBL5410324)
Affinity DataIC50: 0.25nMAssay Description:Displacement of [35S]MK-0677 from human GHSR1a expressed in HEK293 cell membrane by filter binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626070(CHEMBL5402226)
Affinity DataIC50: 0.920nMAssay Description:Displacement of his-tagged [125I]-ghrelin from eYFP-labelled GHSR1a (unknown origin) transfected in HEK293 cells incubated for 20 mins by radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626071(CHEMBL5411243)
Affinity DataIC50: 1.20nMAssay Description:Displacement of his-tagged [125I]-ghrelin from eYFP-labelled GHSR1a (unknown origin) transfected in HEK293 cells incubated for 20 mins by radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626072(CHEMBL5416334)
Affinity DataIC50: 1.40nMAssay Description:Displacement of his-tagged [125I]-ghrelin from eYFP-labelled GHSR1a (unknown origin) transfected in HEK293 cells incubated for 20 mins by radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626069(CHEMBL5426545)
Affinity DataIC50: 2.30nMAssay Description:Displacement of his-tagged [125I]-ghrelin from eYFP-labelled GHSR1a (unknown origin) transfected in HEK293 cells incubated for 20 mins by radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626073(CHEMBL5414374)
Affinity DataIC50: 4nMAssay Description:Displacement of his-tagged [125I]-ghrelin from eYFP-labelled GHSR1a (unknown origin) transfected in HEK293 cells incubated for 20 mins by radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626074(CHEMBL5438862)
Affinity DataIC50: 4.90nMAssay Description:Displacement of his-tagged [125I]-ghrelin from eYFP-labelled GHSR1a (unknown origin) transfected in HEK293 cells incubated for 20 mins by radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626066(CHEMBL5410324)
Affinity DataIC50: 7.60nMAssay Description:Displacement of his-tagged [125I]-ghrelin from eYFP-labelled GHSR1a (unknown origin) transfected in HEK293 cells incubated for 20 mins by radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626068(CHEMBL5411633)
Affinity DataIC50: 7.90nMAssay Description:Displacement of [125I]ghrelin from GHSR1a in HEK293 cells by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Western Ontario

Curated by ChEMBL
LigandPNGBDBM50626065(CHEMBL5402635)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [35S]MK-0677 from human GHSR1a expressed in HEK293 cell membrane by filter binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed