Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50020530
TargetAdenosine receptor A2a(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630906(CHEMBL5430246)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]-SCH58261 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2a(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630909(CHEMBL5413371)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-SCH58261 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2a(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630910(CHEMBL5438060)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]-SCH58261 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630911(CHEMBL5426527)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to recombinant human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2a(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630907(CHEMBL5413330)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [3H]-SCH58261 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2a(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630908(CHEMBL5426841)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]-SCH58261 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2a(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630911(CHEMBL5426527)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]-SCH58261 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630909(CHEMBL5413371)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to recombinant human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630910(CHEMBL5438060)
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to recombinant human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630906(CHEMBL5430246)
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to recombinant human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630907(CHEMBL5413330)
Affinity DataIC50: 3.10nMAssay Description:Binding affinity to recombinant human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAdenosine receptor A2b(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50630908(CHEMBL5426841)
Affinity DataIC50: 3.30nMAssay Description:Binding affinity to recombinant human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 15 to 30 mins by Topcount scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed