Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50020024
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 990nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of porcine PDHc E1-subunit incubated for 30 mins followed by pyruvate addition in presence of thiamine pyrophosphate by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 105nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
TargetPyruvate dehydrogenase E1 component subunit alpha, somatic form, mitochondrial(Pig)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Binding affinity to porcine PDHc E1-subunit assessed as inhibition constant incubated for 30 mins followed by pyruvate addition by microplate reader ...More data for this Ligand-Target Pair
Ligand InfoSimilars
