Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50019759
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50622730(CHEMBL5413288)
Affinity DataKd:  154nMAssay Description:Binding affinity to wild type Nur77 ligand binding domain (unknown origin) assessed as decrease in fluorescence intensity incubated for 30 secs by fl...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50622730(CHEMBL5413288)
Affinity DataKd:  91nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50622731(CHEMBL5398492)
Affinity DataKd:  354nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565399(CHEMBL4795792)
Affinity DataKd:  1.34E+3nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50622732(CHEMBL5419963)
Affinity DataKd:  1.17E+3nMAssay Description:Binding affinity to His-tagged Nur77 ligand binding domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed