Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50020539
Affinity DataEC50: 1.96E+4nMAssay Description:Positive allosteric modulation of recombinant human IDOL transfected in mouse P1.HTR cells assessed as increase in Kyn production incubated for 24 hr...More data for this Ligand-Target Pair
Affinity DataEC50: 4.10E+3nMAssay Description:Activation of OGG1 (unknown origin) by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+3nMAssay Description:Activation of OGG1 (unknown origin) by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.60E+3nMAssay Description:Activation of OGG1 (unknown origin) by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Activation of OGG1 (unknown origin) by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 780nMAssay Description:Activation of OGG1 (unknown origin) by fluorescence-based assayMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataEC50: 37nMAssay Description:Activation of NAMPT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 6.00E+3nMAssay Description:Activation of NAMPT (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 370nMAssay Description:Activation of N-terminal His-tagged human NAMPT-mediated NMN production expressed in Escherichia coli BL21(DE3) cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Activation of 6XHis-FP-rhodamine-tagged full-length mouse LYPLAL1 expressed in Escherichia coli BL21(DE3) cells preincubated for 60 mins followed by ...More data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Activation of 6XHis-FP-rhodamine-tagged full-length human LYPLAL1 expressed in Escherichia coli BL21(DE3) cells preincubated for 60 mins followed by ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+4nMAssay Description:Positive allosteric modulation of recombinant mouse IDOL transfected in mouse P1.HTR cells assessed as increase in Kyn production incubated for 24 hr...More data for this Ligand-Target Pair
Affinity DataEC50: 2.01E+4nMAssay Description:Activation of recombinant human ACE2 using McaAPK(Dnp)-OH as substrate preincubated for 15 mins followed by substrate addition spectra max Gemini M5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Activation of PDE4D5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Activation of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+6nMAssay Description:Activation of G6PD dimerization in lymphocytes isolated from G6PD-deficient patient carrying canton variant expressed in Escherichia coli C43(DE3) ce...More data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:Activation of G6PD (unknown origin) expressed in Escherichia coli C43(DE3) cells using G6P as substrate in presence of NADP+ by resazurin dye-based a...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Nebraska
Curated by ChEMBL
University of Nebraska
Curated by ChEMBL
Affinity DataEC50: 1.10E+5nMAssay Description:Activation of CLpP (unknown origin)More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Nebraska
Curated by ChEMBL
University of Nebraska
Curated by ChEMBL
Affinity DataEC50: 440nMAssay Description:Binding affinity to CLpP (unknown origin)More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Nebraska
Curated by ChEMBL
University of Nebraska
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Activation of recombinant human CLpP using casein-FITC as substrate preincubated for 30 mins followed by substrate addition by spectra max i3x fluore...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
University of Nebraska
Curated by ChEMBL
University of Nebraska
Curated by ChEMBL
Affinity DataEC50: 1.25E+4nMAssay Description:Activation of recombinant human CLpP using Ac-WLA-AMC as substrate preincubated for 60 mins followed by substrate addition by fluorescence based assa...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Human)
University of Nebraska
Curated by ChEMBL
University of Nebraska
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Activation of CPT-1 in digitonin-permeabilized human MCF7 cells preincubated for 2 hrs followed by digitonin addition for 6 mins by liquid scintillat...More data for this Ligand-Target Pair
Affinity DataEC50: 1.95E+4nMAssay Description:Activation of recombinant human ACE2 using McaAPK(Dnp)-OH as substrate preincubated for 15 mins followed by substrate addition spectra max Gemini M5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 8.04E+3nMAssay Description:Activation of recombinant human ACE2 using McaAPK(Dnp)-OH as substrate preincubated for 15 mins followed by substrate addition spectra max Gemini M5 ...More data for this Ligand-Target Pair
