Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50020461
Affinity DataKd: 410nMAssay Description:Binding affinity to N-terminal his6-tagged 53BP1 tandem tudor domain (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) pLysS ...More data for this Ligand-Target Pair
Affinity DataKd: 850nMAssay Description:Binding affinity to N-terminal his6-tagged 53BP1 tandem tudor domain (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) pLysS ...More data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity to N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) pLysS competent cells asse...More data for this Ligand-Target Pair
Affinity DataKd: 790nMAssay Description:Binding affinity to N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) pLysS competent cells asse...More data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Antagonist activity at nanoluc-tagged 53BP1 tandem tudor domain (unknown origin) transfected in HEK293T cells assessed as inhibition of 53BP1-H4 pept...More data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Antagonist activity at nanoluc-tagged 53BP1 tandem tudor domain (unknown origin) transfected in HEK293T cells assessed as inhibition of 53BP1-H4 pept...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+4nMAssay Description:Displacement of Biotin-p53K381acK382me2 from N-terminal his6-tagged 53BP1 (1484 to 1603 residues) (unknown origin) expressed in Rosetta2 BL21 (DE3) p...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at nanoluc-tagged 53BP1 tandem tudor domain (unknown origin) transfected in HEK293T cells assessed as inhibition of 53BP1-H4 pept...More data for this Ligand-Target Pair
TargetM-phase phosphoprotein 8(Homo sapiens)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from MPP8 chromodomain (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetM-phase phosphoprotein 8(Homo sapiens)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from MPP8 chromodomain (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetChromodomain Y-like protein 2(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from CDYL2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetChromodomain Y-like protein 2(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from CDYL2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetChromobox protein homolog 2(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from CBX2 chromodomain (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetChromobox protein homolog 2(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from CBX2 chromodomain (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from PHF19 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from PHF19 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase UHRF1(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of Biotin-p53K381acK382me2 from UHRF1 tandem tudor domain (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
