Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50020360
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629252(CHEMBL5435296)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629253(CHEBI:81892 | Brodifacoum | BRODIFACOUM)
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629247(CHEMBL5436380)
Affinity DataIC50: 498nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629246(CHEMBL5433796)
Affinity DataIC50: 527nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629245(CHEMBL5432023)
Affinity DataIC50: 643nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629250(CHEMBL5403819)
Affinity DataIC50: 873nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50343352(2-hydroxy-3-(3-oxo-1-phenylbutyl)-4H-chromen-4-one...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629244(CHEMBL5404461)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629248(CHEMBL5434421)
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629249(CHEMBL5396437)
Affinity DataIC50: 5.54E+3nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629254(Warfarin alcohol | WARFARIN ALCOHOL)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629251(CHEMBL5424000)
Affinity DataIC50: 2.39E+4nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50629255(Isoprenylcoumarin | ISOPRENYLCOUMARIN)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of recombinant human wild-type VKORC1 expressed in Pichia pastoris membrane incubated for 30 mins in presence of presence of dithiothreito...More data for this Ligand-Target Pair
In DepthDetails
PubMed