Compile Data Set for Download or QSAR
Report error Found 89 Enz. Inhib. hit(s) with all data for entry = 50020212
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627754(CHEMBL5422782)
Affinity DataIC50: 50nMAssay Description:Inhibition of AspH (unknown origin) by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627752(CHEMBL5430087)
Affinity DataIC50: 110nMAssay Description:Inhibition of AspH (unknown origin) by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627747(CHEMBL5429223)
Affinity DataIC50: 280nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM26113(pyridine-2,4-dicarboxylic acid | cid_10365 | pyrid...)
Affinity DataIC50: 300nMAssay Description:Inhibition of his6-tagged human recombinant KDM4E using K9me3 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627735(CHEMBL5419332)
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627732(CHEMBL5425339)
Affinity DataIC50: 400nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627739(CHEMBL5396670)
Affinity DataIC50: 400nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627736(CHEMBL5408048)
Affinity DataIC50: 400nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627732(CHEMBL5425339)
Affinity DataIC50: 500nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM26113(pyridine-2,4-dicarboxylic acid | cid_10365 | pyrid...)
Affinity DataIC50: 500nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant JMJD5 (183 to 416 residues) using RPS6 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627738(CHEMBL5407378)
Affinity DataIC50: 500nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627745(CHEMBL5415306)
Affinity DataIC50: 580nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627737(CHEMBL5423565)
Affinity DataIC50: 700nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627741(CHEMBL5408058)
Affinity DataIC50: 700nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627740(CHEMBL5428941)
Affinity DataIC50: 700nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627734(CHEMBL5402035)
Affinity DataIC50: 900nMAssay Description:Inhibition of N-terminal his6-tagged-thioredoxin-tagged human recombinant JMJD5 expressed in Escherichia coli using RPS6 as substrate by SPE-MS analy...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627740(CHEMBL5428941)
Affinity DataIC50: 900nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627747(CHEMBL5429223)
Affinity DataIC50: 990nMAssay Description:Inhibition of human recombinant KDM4E using biotinylated-H3K9me3 peptide as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627738(CHEMBL5407378)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627748(CHEMBL5429166)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627752(CHEMBL5430087)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of KDM4E (unknown origin) by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627754(CHEMBL5422782)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of KDM4E (unknown origin) by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627733(CHEMBL5434665)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627746(CHEMBL5423241)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627735(CHEMBL5419332)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627739(CHEMBL5396670)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627743(CHEMBL5414235)
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of human recombinant KDM4E using biotinylated-H3K9me3 peptide as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627745(CHEMBL5415306)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition of human recombinant KDM4E using biotinylated-H3K9me3 peptide as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627737(CHEMBL5423565)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627734(CHEMBL5402035)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627747(CHEMBL5429223)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant JMJD5 (183 to 416 residues) using RPS6 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627732(CHEMBL5425339)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant KDM4E expressed in Escherichia coli using K9me3 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627737(CHEMBL5423565)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant KDM4E expressed in Escherichia coli using K9me3 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627735(CHEMBL5419332)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant KDM4E expressed in Escherichia coli using K9me3 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627748(CHEMBL5429166)
Affinity DataIC50: 3.69E+3nMAssay Description:Inhibition of human recombinant KDM4E using biotinylated-H3K9me3 peptide as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627743(CHEMBL5414235)
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627755(CHEMBL5425377)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of AspH (unknown origin) by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627754(CHEMBL5422782)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant JMJD5 (183 to 416 residues) using RPS6 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627749(CHEMBL5401915)
Affinity DataIC50: 5.71E+3nMAssay Description:Inhibition of human recombinant KDM4E using biotinylated-H3K9me3 peptide as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627745(CHEMBL5415306)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant JMJD5 (183 to 416 residues) using RPS6 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627736(CHEMBL5408048)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627733(CHEMBL5434665)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant KDM4E expressed in Escherichia coli using K9me3 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysine-specific demethylase 4E(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627738(CHEMBL5407378)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant KDM4E expressed in Escherichia coli using K9me3 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627748(CHEMBL5429166)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant JMJD5 (183 to 416 residues) using RPS6 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627749(CHEMBL5401915)
Affinity DataIC50: 7.66E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627741(CHEMBL5408058)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of N-terminal his6-tagged AspH (315 to 758 residues) (unknown origin) expressed in Escherichia coli by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627743(CHEMBL5414235)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant JMJD5 (183 to 416 residues) using RPS6 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBifunctional peptidase and arginyl-hydroxylase JMJD5(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627746(CHEMBL5423241)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant JMJD5 (183 to 416 residues) using RPS6 as substrate by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627751(CHEMBL5438950)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAspartyl/asparaginyl beta-hydroxylase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50627750(CHEMBL5414033)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of N-terminal his6-tagged human recombinant AspH (315 to 758 residues) expressed in Escherichia coli BL21 (DE3) cells by SPE-MS analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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