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Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50019302
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617852(CHEMBL5400665)
Affinity DataIC50: 21nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617857(CHEMBL5409784)
Affinity DataIC50: 57nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617845(CHEMBL5423121)
Affinity DataIC50: 72nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617843(CHEMBL5403672)
Affinity DataIC50: 90nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617847(CHEMBL5406504)
Affinity DataIC50: 90nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617851(CHEMBL5420904)
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617852(CHEMBL5400665)
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activity using relaxed pBR322 DNA as substrate preincubated for 5 mins followed by enzyme addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617848(CHEMBL5424692)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617854(CHEMBL5422268)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617856(CHEMBL5435353)
Affinity DataIC50: 160nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617842(CHEMBL5404831)
Affinity DataIC50: 160nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617850(CHEMBL5410417)
Affinity DataIC50: 180nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617858(CHEMBL5424981)
Affinity DataIC50: 190nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617849(CHEMBL5405573)
Affinity DataIC50: 230nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617855(CHEMBL5430363)
Affinity DataIC50: 250nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617853(CHEMBL5409273)
Affinity DataIC50: 270nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617844(CHEMBL5395093)
Affinity DataIC50: 290nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617846(CHEMBL5422850)
Affinity DataIC50: 580nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617852(CHEMBL5400665)
Affinity DataIC50: 900nMAssay Description:Inhibition of human ERG expressed in CHO cells by automated path clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetDNA topoisomerase 2-alpha(Human)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandPNGBDBM50617852(CHEMBL5400665)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 alpha decatenation activity using kDNA as substrate preincubated for 5 mins followed by enzyme addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed