Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50019745
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622666(CHEMBL5432498)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase SUV39H1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human SUV39H1 using Biotin-tagged histone H3 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622650(CHEMBL5423030)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase, H3 lysine-79 specific(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human DOT1L using chicken nucleosome and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622673(CHEMBL5429971)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622667(CHEMBL5411566)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase SMYD3(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human SMYD3 using biotin-tagged MAP3K2 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 9(Homo sapiens)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human PRMT9 using biotin-tagged SAP145 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human PRMT3 using biotin-tagged Histone H4 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetRNA 5'-monophosphate methyltransferase(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human BCDIN3D using biotin-tagged microRNA-145 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622670(CHEMBL5423901)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622657(CHEMBL5407297)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622668(CHEMBL5418908)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622667(CHEMBL5411566)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human GLP using biotin-tagged Histone H3 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622652(CHEMBL5403341)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622651(CHEMBL5416060)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human PRMT1 using biotin-tagged Histone H4 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human MLL1 using biotin-tagged Histone H3 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622655(CHEMBL5407039)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622648(CHEMBL5401536)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622669(CHEMBL5416515)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622654(CHEMBL5437795)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622656(CHEMBL5402316)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human GLP using biotin-tagged Histone H3 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622653(CHEMBL5432737)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622667(CHEMBL5411566)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human G9a using biotin-tagged Histone H3 and 3H-SAM as substrate incubated for 1 hrs by TopCount scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622658(CHEMBL5425227)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622672(CHEMBL5436990)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622671(CHEMBL5405564)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622649(CHEMBL5426089)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622659(CHEMBL5436474)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622660(CHEMBL5399052)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622662(CHEMBL5407441)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622663(CHEMBL5416105)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622664(CHEMBL5432888)
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622665(CHEMBL5394168)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50622661(CHEMBL5435740)
Affinity DataIC50: 3.41E+5nMAssay Description:Inhibition of N-terminal 6His/SUMO-tagged SARS-CoV-2 NSP14 expressed in Escherichia coli Rosetta 2 (DE3) PlysS cells using 5'GpppACCCCCCCCC-Biotin 3'...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed