Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50019743
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50520653(CHEMBL4555209)
Affinity DataKd:  180nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622647(CHEMBL5406183)
Affinity DataKd:  210nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622646(CHEMBL5409305)
Affinity DataKd:  240nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622645(CHEMBL5421103)
Affinity DataKd:  71nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50520653(CHEMBL4555209)
Affinity DataKd:  94nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622647(CHEMBL5406183)
Affinity DataKd:  170nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622646(CHEMBL5409305)
Affinity DataKd:  66nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622645(CHEMBL5421103)
Affinity DataKd:  32nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50520653(CHEMBL4555209)
Affinity DataKd:  35nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622647(CHEMBL5406183)
Affinity DataKd:  26nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622646(CHEMBL5409305)
Affinity DataKd:  26nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622645(CHEMBL5421103)
Affinity DataKd:  160nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50520653(CHEMBL4555209)
Affinity DataKd:  120nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622647(CHEMBL5406183)
Affinity DataKd:  14nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622646(CHEMBL5409305)
Affinity DataKd:  46nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622645(CHEMBL5421103)
Affinity DataKd:  93nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50520653(CHEMBL4555209)
Affinity DataKd:  73nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622647(CHEMBL5406183)
Affinity DataKd:  110nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622646(CHEMBL5409305)
Affinity DataKd:  230nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622645(CHEMBL5421103)
Affinity DataKd:  350nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50520653(CHEMBL4555209)
Affinity DataKd:  680nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622647(CHEMBL5406183)
Affinity DataKd:  8.30nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622646(CHEMBL5409305)
Affinity DataKd:  39nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622645(CHEMBL5421103)
Affinity DataKd:  140nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) assessed as dissociation constant measured for 1200 sec by bio-layer interferometry strepta...More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed