Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50019582
TargetReplicase polyprotein 1ab(2019-nCoV)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM420296(med.21724, Compound 61 | peptidomimetic aldehydes ...)
Affinity DataEC50:  260nMAssay Description:Inhibition of SARS-CoV-2 Main ProteaseMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50619399(CHEMBL5404334)
Affinity DataEC50:  36nMAssay Description:Inhibition of SARS-CoV-2 Main protease expressed in Escherichia coli BL21 (DE3) incubated for 1 hr by affinity chromatography methodMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAngiotensin-converting enzyme 2(Human)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50423643(CEPHARANTHINE)
Affinity DataEC50:  350nMAssay Description:Inhibition of ACE2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50620682(CHEMBL513181 | Ro-9187)
Affinity DataEC50:  0.0300nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50620683(CHEMBL5398494)
Affinity DataEC50:  0.0300nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM60986(cid_16129778 | MLS001335996 | SMR000857330 | TANNI...)
Affinity DataEC50:  585nMAssay Description:Inhibition of N-terminal His6-tagged recombinant full length SARS-CoV-2 3CLpro expressed in Escherichia coli BL21(DE3) using MCA-AVLQSGFR-Lys(Dnp)-Ly...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1a(SARS-CoV)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM60986(cid_16129778 | MLS001335996 | SMR000857330 | TANNI...)
Affinity DataEC50:  8.31E+3nMAssay Description:Inhibition of SARS-CoV 3CLproMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50619399(CHEMBL5404334)
Affinity DataIC50: 120nMAssay Description:Inhibition of SARS-CoV-2 MPro using Dabcyl-KTSAVLQSGFRKME-Edans as substrate preincubated for 5 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50620682(CHEMBL513181 | Ro-9187)
Affinity DataIC50: 171nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50619399(CHEMBL5404334)
Affinity DataIC50: 990nMAssay Description:Inhibition of SARS-CoV-2 PLproMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus type 1)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50530022(CHEMBL438605 | 2''-C-Mecytosine | 2''-C-Methylcyti...)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase associated RNA-dependent DNA polymeraseMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50620682(CHEMBL513181 | Ro-9187)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of Hepatitis C virus NS5B polymeraseMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Qufu Normal University

Curated by ChEMBL
LigandPNGBDBM50620684(4'-AZIDOCYTIDINE | 4'-azidocytidine | R-1479)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails
PubMed