Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50018857
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613254(CHEMBL5271824)
Affinity DataKd:  4.20E+5nMAssay Description:Binding affinity to Escherichia coli TrmD by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613255(CHEMBL5283966)
Affinity DataKd:  2.60E+5nMAssay Description:Binding affinity to Escherichia coli TrmD by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM225673(GTC000445A)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to Escherichia coli TrmD by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613268(CHEMBL5275681)
Affinity DataIC50: 9nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613266(CHEMBL5268562)
Affinity DataIC50: 11nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613282(CHEMBL5270264)
Affinity DataIC50: 13nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613267(CHEMBL5276443)
Affinity DataIC50: 27nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613281(CHEMBL5270195)
Affinity DataIC50: 36nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613279(CHEMBL5290255)
Affinity DataIC50: 37nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613283(CHEMBL5271729)
Affinity DataIC50: 38nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613280(CHEMBL5276347)
Affinity DataIC50: 39nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613269(CHEMBL5291180)
Affinity DataIC50: 50nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613284(CHEMBL5269867)
Affinity DataIC50: 96nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM225684(GTC000457A)
Affinity DataIC50: 110nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613285(CHEMBL5277663)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613270(CHEMBL5288117)
Affinity DataIC50: 130nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613257(CHEMBL5268458)
Affinity DataIC50: 140nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613265(CHEMBL5279532)
Affinity DataIC50: 270nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613260(CHEMBL5289815)
Affinity DataIC50: 310nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613278(CHEMBL5287055)
Affinity DataIC50: 310nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613277(CHEMBL5288124)
Affinity DataIC50: 800nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613276(CHEMBL5274574)
Affinity DataIC50: 830nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613262(CHEMBL5283911)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613258(CHEMBL5268916)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613272(CHEMBL5281871)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613264(CHEMBL5283956)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613259(CHEMBL5290159)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM225672(GTC000444A)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613274(CHEMBL5266230)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613275(CHEMBL5266578)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613261(CHEMBL5267738)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613271(CHEMBL5268413)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM225673(GTC000445A)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613263(CHEMBL5271522)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613273(CHEMBL5287635)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613254(CHEMBL5271824)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM93020(Indole-5-carboxamide)
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613255(CHEMBL5283966)
Affinity DataIC50: 3.20E+5nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106190(4-Amino-benzamide | CHEMBL332444)
Affinity DataIC50: 6.70E+5nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613256(CHEMBL5281955)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed