Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50019698
TargetAlpha-2B adrenergic receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621980(ORM-13070 C-11 | 11c-orm-13070 | Orm-13070 c-11 | ...)
Affinity DataKd:  23nMAssay Description:Binding affinity to alpha2B receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621980(ORM-13070 C-11 | 11c-orm-13070 | Orm-13070 c-11 | ...)
Affinity DataKd:  3.80nMAssay Description:Binding affinity to alpha2C receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621980(ORM-13070 C-11 | 11c-orm-13070 | Orm-13070 c-11 | ...)
Affinity DataKd:  109nMAssay Description:Binding affinity to alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50358166(CHEMBL1921842)
Affinity DataKd:  0.0280nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50049750(CHEMBL59986 | (S)-3-(azetidin-2-ylmethoxy)pyridine...)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity to nACh alpha4beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMu-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataKi:  0.0510nMAssay Description:Binding affinity to mu-opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621981(CHEMBL5412811)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-13-ox...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to delta opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMu-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-13-ox...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to mu-opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621977(CHEMBL5404473)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621978(CHEMBL5428920)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621984(CHEMBL5404578)
Affinity DataKi:  0.360nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621979(CHEMBL5405248)
Affinity DataKi:  0.430nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621983(CHEMBL5438932)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621985(CHEMBL5430462)
Affinity DataKi:  0.670nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50358166(CHEMBL1921842)
Affinity DataKi:  0.720nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621982(CHEMBL5423438)
Affinity DataKi:  0.950nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM26267(RO-154513 | Ro15-4513 | ethyl 12-azido-8-methyl-9-...)
Affinity DataKi:  7nMAssay Description:Binding affinity to GABAa alpha2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM26267(RO-154513 | Ro15-4513 | ethyl 12-azido-8-methyl-9-...)
Affinity DataKi:  7nMAssay Description:Binding affinity to GABAa alpha3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM26267(RO-154513 | Ro15-4513 | ethyl 12-azido-8-methyl-9-...)
Affinity DataKi:  7nMAssay Description:Binding affinity to GABAa alpha1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50296722(p-tolyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylat...)
Affinity DataKi:  14nMAssay Description:Binding affinity to human nACh alpha7 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50296722(p-tolyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylat...)
Affinity DataKi:  22nMAssay Description:Binding affinity to rat nACh alpha7 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMu-type opioid receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50358166(CHEMBL1921842)
Affinity DataKi:  26nMAssay Description:Binding affinity to mu-opioid receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621975(CHEMBL5405359)
Affinity DataKi:  52nMAssay Description:Binding affinity to GluN1/GluN2A receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621986(CHEMBL5404069)
Affinity DataKi:  77nMAssay Description:Binding affinity to nACh alpha6beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50006613(CHEMBL3235480)
Affinity DataKi:  562nMAssay Description:Binding affinity to nACh alpha7 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621974(CHEMBL5418750)
Affinity DataKi:  7.20E+3nMAssay Description:Binding affinity to GluN1/GluN2A receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50433471(CHEMBL2380802)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to nACh alpha4beta2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621976(CHEMBL5411552)
Affinity DataKi:  1.03E+4nMAssay Description:Binding affinity to GluN1/GluN2A receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed