Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50019535
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
3D Structure (crystal)TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
East China University of Science & Technology
Curated by ChEMBL
East China University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of total HDAC in human HUVEC cells using Boc-Lys(Ac)-AMC as substrate preincubated for 12 hrs followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of full-length recombinant human HDAC1 (1 to 482 residues) expressed in baculovirus infected insect cells using Ac-Leu-Gly-Lys(Tfa)-AMC as...More data for this Ligand-Target Pair
