Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50020699
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataKd: 5.20E+3nMAssay Description:Binding affinity to CM5 sensor chip immobilized C-terminal FLAG tagged full length human HAT1/Rbap46 assessed as dissociation constant by SPR analysi...More data for this Ligand-Target Pair
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and 4-pentynoyl...More data for this Ligand-Target Pair
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and 4-pentynoyl...More data for this Ligand-Target Pair
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and acetyl-CoA ...More data for this Ligand-Target Pair
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and 4-pentynoyl...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 6.26E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and 4-pentynoyl...More data for this Ligand-Target Pair
Affinity DataIC50: 7.43E+4nMAssay Description:Inhibition of human p300 incubated for 20 mins followed by 3H-Acetyl CoA addition and measured after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.48E+4nMAssay Description:Inhibition of human MYST2 incubated for 20 mins followed by 3H-Acetyl CoA addition and measured after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.04E+4nMAssay Description:Inhibition of human CBP incubated for 20 mins followed by 3H-Acetyl CoA addition and measured after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human KAT5 incubated for 20 mins followed by 3H-Acetyl CoA addition and measured after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human MYST4 incubated for 20 mins followed by 3H-Acetyl CoA addition and measured after 30 minsMore data for this Ligand-Target Pair
