Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50019002
TargetG-protein coupled bile acid receptor 1(Mouse)
Genentech

Curated by ChEMBL
LigandPNGBDBM50562016(CHEMBL4789628)
Affinity DataEC50:  62nMAssay Description:Inhibition of mouse TGR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Genentech

Curated by ChEMBL
LigandPNGBDBM50614537(CHEMBL5275304)
Affinity DataEC50:  17nMAssay Description:Inhibition of mouse TGR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Genentech

Curated by ChEMBL
LigandPNGBDBM50614538(CHEMBL5286836)
Affinity DataEC50:  0.710nMAssay Description:Inhibition of mouse TGR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50140282(CHEMBL363392 | CHEMBL17879 | 1-{4-[4-((4R,5R)-3,3-...)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of human IBATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetSodium/hydrogen exchanger 3(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM381682(US10272079, Compound 005 | US10272079, Compound 39)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human NHE3More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Mouse)
Genentech

Curated by ChEMBL
LigandPNGBDBM50614537(CHEMBL5275304)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of mouse DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed