Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50019187
TargetSodium/glucose cotransporter 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50386885(CANAGLIFLOZIN HYDRATE | CANAGLIFLOZIN | US10752604...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human SGLT2 by liquid scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP-4 (unknown origin) incubated for 30 mins in presence of substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of voltage dependent L-type calcium channel in rat A7R5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50616349(CHEMBL5414025)
Affinity DataIC50: 4.48E+3nMAssay Description:Inhibition of alpha glucosidase (unknown origin) measured after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of alpha glucosidase (unknown origin) measured after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50616349(CHEMBL5414025)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of voltage dependent L-type calcium channel in rat A7R5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50616349(CHEMBL5414025)
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibition of DPP-4 (unknown origin) incubated for 30 mins in presence of substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSodium/glucose cotransporter 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50616349(CHEMBL5414025)
Affinity DataIC50: 4.11E+5nMAssay Description:Inhibition of human SGLT2 by liquid scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed