Report error Found 149 Enz. Inhib. hit(s) with all data for entry = 50019167
Affinity DataEC50: 0.880nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 3.10nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 204nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 0.880nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 228nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 236nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 3.90nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 0.890nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 5.20nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 3.90nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid scinti...More data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Binding affinity to mouse kappa opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid sci...More data for this Ligand-Target Pair
Affinity DataEC50: 6.70nMAssay Description:Binding affinity to mouse kappa opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid sci...More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Binding affinity to human delta opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid sci...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Binding affinity to human delta opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding incubated for 1.5 hrs by liquid sci...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 0.0210nMAssay Description:Inhibition of human ERG expressed in CHO-K1 cells with holding potential of -80 mV by automated patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 0.0290nMAssay Description:Inhibition of human ERG expressed in CHO-K1 cells with holding potential of -80 mV by automated patch clamp assayMore data for this Ligand-Target Pair
3D Structure (crystal)TargetPotassium voltage-gated channel subfamily H member 2(Human)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inhibition of human ERG expressed in CHO-K1 cells with holding potential of -80 mV by automated patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at mouse mu opioid receptor expressed in CHO cells co-expressing Gqi5 assessed as inhibition of DAMGO induced increase in intrace...More data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Antagonist activity at mouse mu opioid receptor expressed in CHO cells co-expressing Gqi5 assessed as inhibition of DAMGO induced increase in intrace...More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as inhibition constant incubated for 1.5 hrs by competitive radi...More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as inhibition constant incubated for 1.5 hrs by competitive radi...More data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as inhibition constant incubated for 1.5 hrs by competitive radi...More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as inhibition constant incubated for 1.5 hrs by competitive radi...More data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as inhibition constant incubated for 1.5 hrs by competitive radi...More data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cell membrane assessed as inhibition constant incubated for 1.5 hrs by competitive radi...More data for this Ligand-Target Pair
