Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50019507
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619887(CHEMBL5423610)
Affinity DataIC50: 800nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619881(CHEMBL5440285)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619886(CHEMBL5424781)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619869(CHEMBL5433468)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619885(CHEMBL5437731)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619876(CHEMBL5433068)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619873(CHEMBL5425282)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619884(CHEMBL5405727)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619875(CHEMBL5417970)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619888(CHEMBL5411202)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544291(CHEMBL4633662)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619870(CHEMBL5408479)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619889(CHEMBL5408314)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619891(CHEMBL5436428)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619874(CHEMBL5439207)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619883(CHEMBL5394652)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619878(CHEMBL5410036)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619877(CHEMBL5439537)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619890(CHEMBL5397042)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619867(CHEMBL5398979)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544291(CHEMBL4633662)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619874(CHEMBL5439207)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619873(CHEMBL5425282)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619872(CHEMBL5406659)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619871(CHEMBL5408083)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619870(CHEMBL5408479)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619869(CHEMBL5433468)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619868(CHEMBL5409326)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of thiazole orange from His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as decrease in fluorescence in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619881(CHEMBL5440285)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of BLM (unknown origin) assessed as ATP hydrolysis using 5'-biotin-labeled duplex forked-DNA as substrate incubated for 10 mins in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619869(CHEMBL5433468)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of BLM (unknown origin) assessed as ATP hydrolysis using 5'-biotin-labeled duplex forked-DNA as substrate incubated for 10 mins in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619886(CHEMBL5424781)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of BLM (unknown origin) assessed as ATP hydrolysis using 5'-biotin-labeled duplex forked-DNA as substrate incubated for 10 mins in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619887(CHEMBL5423610)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of BLM (unknown origin) assessed as ATP hydrolysis using 5'-biotin-labeled duplex forked-DNA as substrate incubated for 10 mins in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544291(CHEMBL4633662)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of BLM (unknown origin) assessed as ATP hydrolysis using 5'-biotin-labeled duplex forked-DNA as substrate incubated for 10 mins in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619872(CHEMBL5406659)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619871(CHEMBL5408083)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619882(CHEMBL5419427)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619880(CHEMBL5430184)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619868(CHEMBL5409326)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619879(CHEMBL5436259)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619867(CHEMBL5398979)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed