Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50018813
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612852(CHEMBL5281857)
Affinity DataKd: >2.10nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612860(CHEMBL5287352)
Affinity DataKd:  425nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612853(CHEMBL5286815)
Affinity DataKd:  640nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612859(CHEMBL5291013)
Affinity DataKd:  442nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612860(CHEMBL5287352)
Affinity DataKd:  1.19E+3nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612859(CHEMBL5291013)
Affinity DataKd:  3.26E+3nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612858(CHEMBL5276189)
Affinity DataKd: >8.5nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612857(CHEMBL5291407)
Affinity DataKd:  9.89E+4nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612856(CHEMBL5287116)
Affinity DataKd: >2.10nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612855(CHEMBL5279125)
Affinity DataKd:  1.89E+4nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612854(CHEMBL5270591)
Affinity DataKd: >1.10nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612853(CHEMBL5286815)
Affinity DataKd:  1.26E+3nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50084655([(S)-1-((S)-1-Formyl-pentylcarbamoyl)-3-methyl-but...)
Affinity DataKd:  1.22E+3nMAssay Description:Binding affinity to C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612860(CHEMBL5287352)
Affinity DataIC50: 2.37E+3nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50084655([(S)-1-((S)-1-Formyl-pentylcarbamoyl)-3-methyl-but...)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612853(CHEMBL5286815)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612859(CHEMBL5291013)
Affinity DataIC50: 6.49E+3nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612855(CHEMBL5279125)
Affinity DataIC50: 3.78E+4nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612858(CHEMBL5276189)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612857(CHEMBL5291407)
Affinity DataIC50: 1.98E+5nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612854(CHEMBL5270591)
Affinity DataIC50: 2.13E+5nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612856(CHEMBL5287116)
Affinity DataIC50: 4.25E+5nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
European Biomedical Research Institute of Salerno (Ebris)

Curated by ChEMBL
LigandPNGBDBM50612852(CHEMBL5281857)
Affinity DataIC50: 4.25E+5nMAssay Description:Inhibition of C-terminal His6-tagged recombinant SARS-CoV-2 MPro transfected in Escherichia coli BL21 (DE3) using Dabcyl-KTSAVLQSGFRKM-E(Edans)-NH2 a...More data for this Ligand-Target Pair
In DepthDetails
PubMed