Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50018060
LigandPNGBDBM50607315(BAY-069)
Affinity DataIC50: 31nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607303(CHEMBL5220763)
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607314(CHEMBL5219349)
Affinity DataIC50: 70nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50607314(CHEMBL5219349)
Affinity DataIC50: 70nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50607314(CHEMBL5219349)
Affinity DataIC50: 90nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50607311(CHEMBL5220953)
Affinity DataIC50: 120nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607300(CHEMBL5218588)
Affinity DataIC50: 145nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607297(CHEMBL5220319)
Affinity DataIC50: 150nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607315(BAY-069)
Affinity DataIC50: 153nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607286(CHEMBL5218805)
Affinity DataIC50: 159nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607294(CHEMBL5220178)
Affinity DataIC50: 162nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607294(CHEMBL5220178)
Affinity DataIC50: 162nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50607304(CHEMBL5219314)
Affinity DataIC50: 180nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607316(CHEMBL5219436)
Affinity DataIC50: 180nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607315(BAY-069)
Affinity DataIC50: 186nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607315(BAY-069)
Affinity DataIC50: 186nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607316(CHEMBL5219436)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607298(CHEMBL5219261)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607301(CHEMBL5220805)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607316(CHEMBL5219436)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607316(CHEMBL5219436)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607316(CHEMBL5219436)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607316(CHEMBL5219436)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607291(CHEMBL5220903)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607314(CHEMBL5219349)
Affinity DataIC50: 270nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607290(CHEMBL5220488)
Affinity DataIC50: 287nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50607314(CHEMBL5219349)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607314(CHEMBL5219349)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607283(CHEMBL5219683)
Affinity DataIC50: 340nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607284(CHEMBL5218519)
Affinity DataIC50: 400nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607292(CHEMBL5219699)
Affinity DataIC50: 413nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607310(CHEMBL5220057)
Affinity DataIC50: 438nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607289(CHEMBL5219137)
Affinity DataIC50: 507nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607288(CHEMBL5220817)
Affinity DataIC50: 554nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50607302(CHEMBL5219393)
Affinity DataIC50: 700nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607296(CHEMBL5219459)
Affinity DataIC50: 723nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607305(CHEMBL5220789)
Affinity DataIC50: 725nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607299(CHEMBL5219673)
Affinity DataIC50: 792nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607281(CHEMBL5218966)
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607318(CHEMBL5220587)
Affinity DataIC50: 850nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607317(CHEMBL5220979)
Affinity DataIC50: 900nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607295(CHEMBL5219169)
Affinity DataIC50: 925nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607285(CHEMBL5219665)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607315(BAY-069)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607315(BAY-069)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607292(CHEMBL5219699)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607286(CHEMBL5218805)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607293(CHEMBL5219930)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607284(CHEMBL5218519)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50607290(CHEMBL5220488)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
Displayed 1 to 50 (of 78 total ) | Next | Last >>
Jump to: