Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50018780
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612500(CHEMBL5287761)
Affinity DataIC50: 580nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612498(CHEMBL5278604)
Affinity DataIC50: 590nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612497(CHEMBL5277503)
Affinity DataIC50: 760nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612494(CHEMBL5289105)
Affinity DataIC50: 790nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612501(CHEMBL5268217)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612496(CHEMBL5267955)
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612495(CHEMBL5278969)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612499(CHEMBL5270889)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of N-terminal his-tagged human recombinant LSD1 using 10-acetyl-3,7-dihydroxyphenoxazine as substrate measured for 30 mins by multiplate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50612500(CHEMBL5287761)
Affinity DataKi:  5.49E+3nMAssay Description:Inhibition of human recombinant LSD1 assessed as inhibition constant by HRP-coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed