Compile Data Set for Download or QSAR
Report error Found 119 Enz. Inhib. hit(s) with all data for entry = 50015999
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591310(CHEMBL5205289)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591307(CHEMBL5198237)
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591308(CHEMBL5177166)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591309(CHEMBL5193531)
Affinity DataIC50: 5.74E+4nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591302(CHEMBL5194237)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591304(CHEMBL5176469)
Affinity DataIC50: 3.27E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591306(CHEMBL5206696)
Affinity DataIC50: 3.27E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591305(CHEMBL5191973)
Affinity DataIC50: 6.69E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591297(CHEMBL5171860)
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591298(CHEMBL5201114)
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591299(CHEMBL5191609)
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591300(CHEMBL5193118)
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591301(CHEMBL5184240)
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591303(CHEMBL5203377)
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM69602(WB-4101 hydrochloride | N-(2,3-dihydro-1,4-benzodi...)
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibition of human recombinant DPP4 using H-Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591297(CHEMBL5171860)
Affinity DataKi:  7.20nMAssay Description:Inhibition of human recombinant CA2 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant CA2 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591297(CHEMBL5171860)
Affinity DataKi:  20nMAssay Description:Inhibition of human recombinant CA9 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 9(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  26nMAssay Description:Inhibition of human recombinant CA9 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 9(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591309(CHEMBL5193531)
Affinity DataKi:  31nMAssay Description:Inhibition of human recombinant CA9 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591308(CHEMBL5177166)
Affinity DataKi:  36nMAssay Description:Inhibition of human recombinant CA2 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591308(CHEMBL5177166)
Affinity DataKi:  43nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  54nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  63nMAssay Description:Inhibition of human recombinant CA5A assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  74nMAssay Description:Inhibition of human recombinant CA4 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 5A, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591297(CHEMBL5171860)
Affinity DataKi:  78nMAssay Description:Inhibition of human recombinant CA5A assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591306(CHEMBL5206696)
Affinity DataKi:  78nMAssay Description:Inhibition of human recombinant CA5A assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591297(CHEMBL5171860)
Affinity DataKi:  85nMAssay Description:Inhibition of human recombinant CA1 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591307(CHEMBL5198237)
Affinity DataKi:  90nMAssay Description:Inhibition of human recombinant CA5A assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591297(CHEMBL5171860)
Affinity DataKi:  90nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591308(CHEMBL5177166)
Affinity DataKi:  94nMAssay Description:Inhibition of human recombinant CA5A assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 9(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591306(CHEMBL5206696)
Affinity DataKi:  111nMAssay Description:Inhibition of human recombinant CA9 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 9(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591308(CHEMBL5177166)
Affinity DataKi:  133nMAssay Description:Inhibition of human recombinant CA9 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591307(CHEMBL5198237)
Affinity DataKi:  155nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591305(CHEMBL5191973)
Affinity DataKi:  183nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591310(CHEMBL5205289)
Affinity DataKi:  232nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591308(CHEMBL5177166)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]-prazosin from human adrenergic alpha1A receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  250nMAssay Description:Inhibition of human recombinant CA1 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 1(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591308(CHEMBL5177166)
Affinity DataKi:  262nMAssay Description:Inhibition of human recombinant CA1 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591297(CHEMBL5171860)
Affinity DataKi:  291nMAssay Description:Inhibition of human recombinant CA4 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 9(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591305(CHEMBL5191973)
Affinity DataKi:  328nMAssay Description:Inhibition of human recombinant CA9 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591306(CHEMBL5206696)
Affinity DataKi:  350nMAssay Description:Inhibition of human recombinant CA2 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591306(CHEMBL5206696)
Affinity DataKi:  387nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591309(CHEMBL5193531)
Affinity DataKi:  410nMAssay Description:Inhibition of human recombinant CA5B assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591309(CHEMBL5193531)
Affinity DataKi:  456nMAssay Description:Inhibition of human recombinant CA5A assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 4(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591309(CHEMBL5193531)
Affinity DataKi:  478nMAssay Description:Inhibition of human recombinant CA4 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591305(CHEMBL5191973)
Affinity DataKi:  659nMAssay Description:Inhibition of human recombinant CA5A assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 9(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591307(CHEMBL5198237)
Affinity DataKi:  745nMAssay Description:Inhibition of human recombinant CA9 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCarbonic anhydrase 2(Human)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50591309(CHEMBL5193531)
Affinity DataKi:  843nMAssay Description:Inhibition of human recombinant CA2 assessed as inhibition constant pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydra...More data for this Ligand-Target Pair
In DepthDetails
PubMed
Displayed 1 to 50 (of 119 total ) | Next | Last >>
Jump to: