Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50015833
TargetBromodomain-containing protein 4(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50573454(CHEMBL4854720)
Affinity DataIC50: 10nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD1 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50573455(CHEMBL4848064)
Affinity DataIC50: 34nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD1 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50590048(CHEMBL5178566)
Affinity DataIC50: 38nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD1 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50573454(CHEMBL4854720)
Affinity DataIC50: 108nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD2 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50573455(CHEMBL4848064)
Affinity DataIC50: 118nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD2 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50590048(CHEMBL5178566)
Affinity DataIC50: 188nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD2 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed