Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50017332
TargetShort transient receptor potential channel 5(Human)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50601265(CHEMBL5177160)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human TRPC5 stably expressed in T-REx-293 cells assessed as increase in calcium flux by Fura-2AM dye based fluorescence plate rea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50601266(CHEMBL5173479)
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at human TRPC5 stably expressed in T-REx-293 cells assessed as increase in calcium flux by Fura-2AM dye based fluorescence plate rea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50601267(ENGLERIN A | CHEBI:72441 | Englerin A)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at human TRPC5 stably expressed in HEK293 cells assessed as increase in calcium flux by Fura-2AM dye based fluorescence plate reader...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed