Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50016200
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50087820(CHEMBL3426797)
Affinity DataEC50:  1.41E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM224018((+)-TAN-67)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human DOR expressed in CHO cells assessed as reduction in ERK1/2 phosphorylation levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50059833(4-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human DOR expressed in CHO cells assessed as reduction in ERK1/2 phosphorylation levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human DOR expressed in CHO cells assessed as reduction in ERK1/2 phosphorylation levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593191(CHEMBL5195022)
Affinity DataEC50:  5.01E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593190(CHEMBL5182141)
Affinity DataEC50:  2.04E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593189(CHEMBL5191568)
Affinity DataEC50:  8.13E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593188(CHEMBL5205658)
Affinity DataEC50:  1.62E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593187(CHEMBL5190988)
Affinity DataEC50:  2.40E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593186(CHEMBL5191793)
Affinity DataEC50:  3.47E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593185(CHEMBL5200037)
Affinity DataEC50:  1.38E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593184(CHEMBL5189216)
Affinity DataEC50:  2.75E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593183(CHEMBL5184328)
Affinity DataEC50:  3.47E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50087826(CHEMBL3426789)
Affinity DataEC50:  3.47E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50087826(CHEMBL3426789)
Affinity DataEC50:  2.34E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593191(CHEMBL5195022)
Affinity DataEC50:  2.04E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593190(CHEMBL5182141)
Affinity DataEC50:  3.55E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593189(CHEMBL5191568)
Affinity DataEC50:  5.75E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593188(CHEMBL5205658)
Affinity DataEC50:  2.34E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593187(CHEMBL5190988)
Affinity DataEC50:  8.32E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593186(CHEMBL5191793)
Affinity DataEC50:  1.62E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593185(CHEMBL5200037)
Affinity DataEC50:  2.19E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593184(CHEMBL5189216)
Affinity DataEC50:  2.75E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593183(CHEMBL5184328)
Affinity DataEC50:  3.47E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50087820(CHEMBL3426797)
Affinity DataEC50:  1.91E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed