Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50018004
Affinity DataEC50: 6.46E+3nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 776nMAssay Description:Positive allosteric modulation of GPR40 (unknown origin)More data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Human)
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of LPAAT-beta (unknown origin) expressed in Xenopus laevis oocytes incubated for 3 minsMore data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Human)
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of LPAAT-beta (unknown origin) expressed in Xenopus laevis oocytes incubated for 3 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of IMPDH2 (unknown origin)More data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Human)
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human LPAAT-beta by cell-free colorimetric assayMore data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Human)
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human LPAAT-beta by cell-free colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of cGAS (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibition of human NOX5More data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of human ENT1 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:Inhibition of human NOX4More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of human NOX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of human NOX3More data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of human ENT1 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human NOX3More data for this Ligand-Target Pair
Affinity DataIC50: 4.36E+3nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-adenosine uptake by liquid sc...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human NOX1More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human NOX1More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human NOX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human ENT1 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of human ENT1 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-adenosine uptake by liquid sc...More data for this Ligand-Target Pair
Affinity DataIC50: 7.71E+4nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.83E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.29E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.54E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.76E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.71E+3nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
