Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50016357
TargetPup--protein ligase(Corynebacterium glutamicum (strain ATCC 13032 / DS...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50594452(SEPANTRONIUM | Sepantronium cation | Sepantronium ...)
Affinity DataEC50:  1.70E+3nMAssay Description:Activation of Corynebacterium glutamicum PafA expressed in Escherichia coli BL-21(DE3) assessed as pup-ylation using Mtb PanB substrate by SDS-PAGE a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetPup--protein ligase(Corynebacterium glutamicum (strain ATCC 13032 / DS...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50594452(SEPANTRONIUM | Sepantronium cation | Sepantronium ...)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of Corynebacterium glutamicum PafA expressed in Escherichia coli BL-21(DE3) assessed as pup-ylation using Mtb KasA substrate by SDS-PAGE a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetPup--protein ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM36880(cid_2406 | SMR000058374 | 2,4-dichloro-6-(3,5-dich...)
Affinity DataIC50: 1.59E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PafA expressed in Escherichia coli BL-21(DE3) assessed as inhibition of pup-ylation using Mtb PanB substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetPup--protein ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50124518((E)-4-[3-(1-adamantyl)-4-hydroxyphenyl]cinnamic ac...)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PafA expressed in Escherichia coli BL-21(DE3) assessed as inhibition of pup-ylation using Mtb PanB substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed