Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50015789
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589556(CHEMBL5207498)
Affinity DataKi:  0.661nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589552(CHEMBL5207290)
Affinity DataKi:  0.676nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589556(CHEMBL5207498)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589546(CHEMBL5172513)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589555(CHEMBL5208506)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589550(CHEMBL5196082)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589554(CHEMBL5205220)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589552(CHEMBL5207290)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589554(CHEMBL5205220)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589551(CHEMBL5195884)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589550(CHEMBL5196082)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589548(CHEMBL5176227)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589549(CHEMBL5175698)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589548(CHEMBL5176227)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589546(CHEMBL5172513)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589553(CHEMBL5185103)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589555(CHEMBL5208506)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589551(CHEMBL5195884)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589553(CHEMBL5185103)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589545(CHEMBL5198830)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50042209(4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  191nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50042209(4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589547(CHEMBL5172969)
Affinity DataKi:  525nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589547(CHEMBL5172969)
Affinity DataKi:  562nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589549(CHEMBL5175698)
Affinity DataKi:  617nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAdenosine receptor A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50589545(CHEMBL5198830)
Affinity DataKi:  955nMAssay Description:Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement a...More data for this Ligand-Target Pair
In DepthDetails
PubMed