Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50016512
Affinity DataKd: 37nMAssay Description:Binding affinity to His6/TEV fused recombinant human BRD4 expressed in bacteria assessed as dissociation constant by isothermal titration calorimetry...More data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Inhibition of PLK1 in thymidine synchronized human HeLa cells using casein as substrate preincubated with compound for 13 hrs followed by substrate a...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of PLK1 PBD (unknown origin) using 5CF-GPMQSpTPLNG-NH2 as substrate preincubated for 30 mins followed by substrate addition and measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant full length human PLK1 using casein as substrate incubated for 40 mins in the presence of [gamma33P]ATP at Km concentration...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Competitive inhibition of 5-carboxyfluorescein-GPMQSpTPLNQ-OH binding to PLK1 PBD (371 to 603 residues) (unknown origin) incubated for 60 mins by flu...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human PLK1 in the presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human PLK2 (65 to 409 resiudes) using casein as substrate incubated for 40 mins in the presence of [gamma33P]ATP at Km conc...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Myc-tagged PLK1 PBD (unknown origin) expressed in HEK293T cells using 5CF-GPMQSpTPLNG-NH2 as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of biotinylated p-T78 peptide binding to human HA-EGFP-PLK1 expressed in HEK293-A cells using TMB as substrate incubated for 1 hrs by ELIS...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human Wee1 in the presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of Myc-tagged PLK1 PBD (unknown origin) expressed in HEK293T cells using 5CF-GPMQSpTPLNG-NH2 as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Competitive inhibition of 5-carboxyfluorescein-GPMQSpTPLNQ-OH binding to PLK1 PBD (371 to 603 residues) (unknown origin) incubated for 60 mins by flu...More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of Myc-tagged PLK2 PBD (unknown origin) expressed in HEK293T cells using 5CF-GPMQTSpTPKNG-NH2 as substrate preincubated for 30 mins follow...More data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Inhibition of Myc-tagged PLK2 PBD (unknown origin) expressed in HEK293T cells using 5CF-GPMQTSpTPKNG-NH2 as substrate preincubated for 30 mins follow...More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of PLK2 PBD (unknown origin) using 5CF-GPMQTSpTPKNG-NH2 as substrate preincubated for 30 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of PLK1 PBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 770nMAssay Description:Inhibition of PLK1 PBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Inhibition of PLK1 PBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inhibition of PLK1 PBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 960nMAssay Description:Inhibition of PLK1 PBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 980nMAssay Description:Inhibition of PLK3 PBD (unknown origin) using 5CF-PLATSpTPKNG-NH2 as substrate preincubated for 30 mins followed by substrate addition and measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 990nMAssay Description:Inhibition of PLK1 PBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of biotin labelled PoloBoxtide binding to GST/His-fused full length PLK1 (unknown origin) expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Myc-tagged PLK3 PBD (unknown origin) expressed in HEK293T cells using 5CF-PLATSpTPKNG-NH2 as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of 5-carboxyfluoresceinGPMQSpTPLNG-OH peptide binding to N-terminal His7-tagged human PLK1 (326 to 603 residues) PBD expressed in Escheric...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of biotinylated PLHSpT peptide binding to n-terminal GST-tagged full length human PLK1 PBD preincubated with compound for 30 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of Myc-tagged PLK3 PBD (unknown origin) expressed in HEK293T cells using 5CF-PLATSpTPKNG-NH2 as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of PLK1 T210D mutant kinase domain (unknown origin) using casein as substrate preincubated for 3 hrs followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of biotinylated p-T78 peptide binding to human HA-EGFP-PLK1 expressed in HEK293-A cells using TMB as substrate incubated for 1 hrs by ELIS...More data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of 5-carboxyfluoresceinGPMQSpTPLNG-OH peptide binding to human PLK1 (326 to 603 residues) PBD expressed in Rosetta BL21 (DE3) cells preinc...More data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of Myc-tagged PLK2 PBD (unknown origin) expressed in HEK293T cells using 5CF-GPMQTSpTPKNG-NH2 as substrate preincubated for 30 mins follow...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of PLK1 (unknown origin) in the presence of ATP by ADP-Glo-kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of PLK1 (unknown origin) in the presence of ATP by ADP-Glo-kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of Myc-tagged PLK3 PBD (unknown origin) expressed in HEK293T cells using 5CF-PLATSpTPKNG-NH2 as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of PLK1 (unknown origin) in the presence of ATP by ADP-Glo-kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of 5-carboxyfluoresceinGPMQSpTPLNG-OH peptide binding to PLK1 (326 to 603 residues) PBD (unknown origin) preincubated for 1 hrs with compo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of 5-carboxyfluorescein-GPMQTSpTPKNG-OH peptide binding to PLK2 (355 to 685 residues) PBD (unknown origin) preincubated for 1 hrs with com...More data for this Ligand-Target Pair
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of 5-carboxyfluoresceinGPMQSpTPLNG-OH peptide binding to human PLK1 (326 to 603 residues) PBD expressed in Rosetta BL21 (DE3) cells preinc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of 5-carboxyfluorescein-GPMQTSpTPKNG-OH peptide binding to C-terminal 6His-tagged human PLK2 (355 to 685 residues) PBD expressed in Rosett...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of biotin labelled PoloBoxtide binding to GST/His-fused full length PLK1 (unknown origin) expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of biotinylated p-T78 peptide binding to human HA-EGFP-PLK1 expressed in HEK293-A cells using TMB as substrate incubated for 1 hrs by ELIS...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of PLK3 (unknown origin) in the presence of ATP by ADP-Glo-kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.82E+4nMAssay Description:Inhibition of 5-carboxyfluoresceinGPMQSpTPLNG-OH peptide binding to PLK1 (326 to 603 residues) PBD (unknown origin) preincubated for 1 hrs with compo...More data for this Ligand-Target Pair
Affinity DataIC50: 5.19E+4nMAssay Description:Inhibition of 5-carboxyfluorescein-GPMQTSpTPKNG-OH peptide binding to PLK2 (355 to 685 residues) PBD (unknown origin) preincubated for 1 hrs with com...More data for this Ligand-Target Pair
Affinity DataIC50: 5.39E+4nMAssay Description:Inhibition of 5-carboxyfluorescein-GPLATSpTPKNG-OH peptide binding to N-terminal MBP-tagged human PLK3 (335 to 646 residues) PBD expressed in Rosetta...More data for this Ligand-Target Pair
Affinity DataIC50: 5.48E+4nMAssay Description:Inhibition of 5-carboxyfluorescein-GPMQTSpTPKNG-OH peptide binding to PLK2 (355 to 685 residues) PBD (unknown origin) preincubated for 1 hrs with com...More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of PLK1 PBD (unknown origin) dependent bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of PLK1 PBD (unknown origin) dependent bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.42E+5nMAssay Description:Inhibition of PLK2 (unknown origin) in the presence of ATP by ADP-Glo-kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.14E+5nMAssay Description:Inhibition of PLK2 (unknown origin) in the presence of ATP by ADP-Glo-kinase assayMore data for this Ligand-Target Pair
