Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50016342
TargetMediator of RNA polymerase II transcription subunit 25(Human)
University of Utah College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50442875(NORSTICTIC ACID)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Med25 transcriptional activation in human MCF-7 cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
Target14 kDa phosphohistidine phosphatase(Human)
University of Utah College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50442875(NORSTICTIC ACID)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails
PubMed
Target14 kDa phosphohistidine phosphatase(Human)
University of Utah College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50056922(cid_73677 | CHEMBL173530 | 1,4-Dihydroxy-10-methox...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails
PubMed
Target14 kDa phosphohistidine phosphatase(Human)
University of Utah College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50239376(ROXARSONE | CHEBI:35817)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails
PubMed
Target14 kDa phosphohistidine phosphatase(Human)
University of Utah College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50240028(Acetarsol | Acetarsone | Gynoplix | S.V.C. | Stova...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails
PubMed
Target14 kDa phosphohistidine phosphatase(Human)
University of Utah College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50442875(NORSTICTIC ACID)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of PHPT1 (unknown origin) assessed as inhibition constant measured up to 100 uM incubated up to 30 mins using DiFMUP as fluorogenic substr...More data for this Ligand-Target Pair
In DepthDetails
PubMed