Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50016123
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50079362(CHEMBL3417009 | US9663465, 9)
Affinity DataIC50: 16nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and by DTNB reagent based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592626(CHEMBL5187324)
Affinity DataIC50: 880nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592624(CHEMBL5208032)
Affinity DataIC50: 990nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592622(CHEMBL5185065)
Affinity DataIC50: 2.59E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592631(CHEMBL5205468)
Affinity DataIC50: 3.45E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592628(CHEMBL5185843)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592625(CHEMBL5203792)
Affinity DataIC50: 3.79E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592622(CHEMBL5185065)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592618(CHEMBL5172343)
Affinity DataIC50: 4.56E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592620(CHEMBL5186394)
Affinity DataIC50: 5.14E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50199522((+-)-HA | (1R,9R)-1-Amino-13-eth-(E)-ylidene-11-me...)
Affinity DataIC50: 5.28E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592629(CHEMBL5186796)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592625(CHEMBL5203792)
Affinity DataIC50: 5.73E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592621(CHEMBL5204734)
Affinity DataIC50: 6.08E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592619(CHEMBL5171192)
Affinity DataIC50: 6.24E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592623(CHEMBL5171010)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592623(CHEMBL5171010)
Affinity DataIC50: 6.66E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592617(CHEMBL5193255)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592616(CHEMBL5186051)
Affinity DataIC50: 8.36E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592615(CHEMBL5196988)
Affinity DataIC50: 9.16E+3nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592615(CHEMBL5196988)
Affinity DataIC50: 9.82E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592621(CHEMBL5204734)
Affinity DataIC50: 9.94E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592627(CHEMBL5171268)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592626(CHEMBL5187324)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592618(CHEMBL5172343)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592629(CHEMBL5186796)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592630(CHEMBL5199425)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592628(CHEMBL5185843)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592620(CHEMBL5186394)
Affinity DataIC50: 2.89E+4nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592619(CHEMBL5171192)
Affinity DataIC50: 2.98E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592617(CHEMBL5193255)
Affinity DataIC50: 2.98E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592631(CHEMBL5205468)
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592627(CHEMBL5171268)
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592630(CHEMBL5199425)
Affinity DataIC50: 3.14E+4nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592616(CHEMBL5186051)
Affinity DataIC50: 4.49E+4nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592624(CHEMBL5208032)
Affinity DataIC50: 4.84E+4nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50199522((+-)-HA | (1R,9R)-1-Amino-13-eth-(E)-ylidene-11-me...)
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of BuChE (unknown origin) using butyrylthiocholine iodide as substrate by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50079362(CHEMBL3417009 | US9663465, 9)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]GR113808 from human 5-HT4 receptor expressed in Chem-1 cell membrane incubated for 60 mins by radiometric scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Hebei University

Curated by ChEMBL
LigandPNGBDBM50592632(CHEMBL5190650)
Affinity DataKi:  312nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by DTNB reagent based spectrophotometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed