Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50016810
LigandPNGBDBM50597411(CHEMBL5171387)
Affinity DataIC50: 2nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 3nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597425(CHEMBL5194202)
Affinity DataIC50: 4nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597424(CHEMBL5187378)
Affinity DataIC50: 4nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597419(CHEMBL5182767)
Affinity DataIC50: 4nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597426(CHEMBL5169449)
Affinity DataIC50: 5nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597406(CHEMBL5207899)
Affinity DataIC50: 5nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597410(CHEMBL5184795)
Affinity DataIC50: 5nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597421(CHEMBL5209068)
Affinity DataIC50: 5nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 6nMAssay Description:Inhibition of GST-tagged human CDK9/Cyclin T1 expressed in Sf9 cells using (YSPTSPS)2KK peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597407(CHEMBL5191136)
Affinity DataIC50: 6nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597423(CHEMBL5183669)
Affinity DataIC50: 6nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597415(CHEMBL5187158)
Affinity DataIC50: 6nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 12(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 7nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597409(CHEMBL5169627)
Affinity DataIC50: 8nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597427(CHEMBL5195127)
Affinity DataIC50: 9nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597414(CHEMBL5176463)
Affinity DataIC50: 11nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597419(CHEMBL5182767)
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged human CDK9/Cyclin T1 expressed in Sf9 cells using (YSPTSPS)2KK peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597418(CHEMBL5179519)
Affinity DataIC50: 12nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597428(CHEMBL5194833)
Affinity DataIC50: 12nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597426(CHEMBL5169449)
Affinity DataIC50: 12nMAssay Description:Inhibition of GST-tagged human CDK9/Cyclin T1 expressed in Sf9 cells using (YSPTSPS)2KK peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 13/Cyclin-K(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597426(CHEMBL5169449)
Affinity DataIC50: 12nMAssay Description:Inhibition of GST-tagged human CDK13/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 18nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597416(CHEMBL5205821)
Affinity DataIC50: 19nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597425(CHEMBL5194202)
Affinity DataIC50: 20nMAssay Description:Inhibition of GST-tagged human CDK9/Cyclin T1 expressed in Sf9 cells using (YSPTSPS)2KK peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 13/Cyclin-K(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 21nMAssay Description:Inhibition of GST-tagged human CDK13/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 13/Cyclin-K(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597425(CHEMBL5194202)
Affinity DataIC50: 22nMAssay Description:Inhibition of GST-tagged human CDK13/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 13/Cyclin-K(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597424(CHEMBL5187378)
Affinity DataIC50: 22nMAssay Description:Inhibition of GST-tagged human CDK13/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597424(CHEMBL5187378)
Affinity DataIC50: 23nMAssay Description:Inhibition of GST-tagged human CDK9/Cyclin T1 expressed in Sf9 cells using (YSPTSPS)2KK peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597403(CHEMBL5208001)
Affinity DataIC50: 24nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597408(CHEMBL5173574)
Affinity DataIC50: 25nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 12(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597426(CHEMBL5169449)
Affinity DataIC50: 29nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597405(CHEMBL5176720)
Affinity DataIC50: 37nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597428(CHEMBL5194833)
Affinity DataIC50: 38nMAssay Description:Inhibition of GST-tagged human CDK9/Cyclin T1 expressed in Sf9 cells using (YSPTSPS)2KK peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597412(CHEMBL5201329)
Affinity DataIC50: 43nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 12(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597424(CHEMBL5187378)
Affinity DataIC50: 50nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597404(CHEMBL5187017)
Affinity DataIC50: 53nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597407(CHEMBL5191136)
Affinity DataIC50: 62nMAssay Description:Inhibition of GST-tagged human CDK9/Cyclin T1 expressed in Sf9 cells using (YSPTSPS)2KK peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 12(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597425(CHEMBL5194202)
Affinity DataIC50: 64nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 13/Cyclin-K(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597419(CHEMBL5182767)
Affinity DataIC50: 67nMAssay Description:Inhibition of GST-tagged human CDK13/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 12(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597419(CHEMBL5182767)
Affinity DataIC50: 73nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597413(CHEMBL5201069)
Affinity DataIC50: 75nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 115nMAssay Description:Inhibition of GST-tagged CDK2/cyclin D1 (unknown origin) expressed in Sf9 cells using RPPTLSPIPHIPR peptide as substrate in presence of ATP and [gamm...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 13/Cyclin-K(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597407(CHEMBL5191136)
Affinity DataIC50: 122nMAssay Description:Inhibition of GST-tagged human CDK13/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 12(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597407(CHEMBL5191136)
Affinity DataIC50: 156nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597402(CHEMBL5171541)
Affinity DataIC50: 256nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 12(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597428(CHEMBL5194833)
Affinity DataIC50: 304nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 13/Cyclin-K(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50597428(CHEMBL5194833)
Affinity DataIC50: 334nMAssay Description:Inhibition of GST-tagged human CDK13/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597420(CHEMBL5198145)
Affinity DataIC50: 464nMAssay Description:Inhibition of His-tagged CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of ATP and [gamma33-P]ATP b...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50597426(CHEMBL5169449)
Affinity DataIC50: 940nMAssay Description:Inhibition of GST-tagged CDK2/cyclin D1 (unknown origin) expressed in Sf9 cells using RPPTLSPIPHIPR peptide as substrate in presence of ATP and [gamm...More data for this Ligand-Target Pair
In DepthDetails
PubMed
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