Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50017903
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605978(CHEMBL2326523)
Affinity DataKd:  1.18E+4nMAssay Description:Binding affinity to human recombinant LC3B assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605979(CHEMBL5180355)
Affinity DataKd:  175nMAssay Description:Binding affinity to human recombinant LC3B assessed as dissociation constant incubated for 30 mins by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605982(CHEMBL5170949)
Affinity DataKd:  993nMAssay Description:Binding affinity to LC3B (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605985(CHEMBL5208126)
Affinity DataIC50: 10nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605986(CHEMBL5195481)
Affinity DataIC50: 10nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605984(CHEMBL5186406)
Affinity DataIC50: 13nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605980(CHEMBL5195612)
Affinity DataIC50: 15nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605981(CHEMBL5190733)
Affinity DataIC50: 19nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605982(CHEMBL5170949)
Affinity DataIC50: 23nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605983(CHEMBL5209227)
Affinity DataIC50: 34nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605977(CHEMBL5191002)
Affinity DataIC50: 85nMAssay Description:Inhibition of human recombinant NAMPT preincubated for 5 mins followed by addition NAMPT measured after 15 mins by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50605977(CHEMBL5191002)
Affinity DataIC50: 85nMAssay Description:Inhibition of NAMPT (unknown origin) measured after 90 mins by measuring fluorescence intensityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed