Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50016742
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596984(CHEMBL5207485)
Affinity DataIC50: 390nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596980(CHEMBL5180404)
Affinity DataIC50: 750nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50568522(CHEMBL4864352)
Affinity DataIC50: 870nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596981(CHEMBL5186476)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596982(CHEMBL5177471)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596975(CHEMBL5184132)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596972(CHEMBL5172654)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596977(CHEMBL5179061)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596974(CHEMBL5175317)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596976(CHEMBL5200476)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596983(CHEMBL5190070)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596973(CHEMBL5206956)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596979(CHEMBL5181710)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596978(CHEMBL5171912)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596985(CHEMBL5170156)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596984(CHEMBL5207485)
Affinity DataKi:  80nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596980(CHEMBL5180404)
Affinity DataKi:  190nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596981(CHEMBL5186476)
Affinity DataKi:  220nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596973(CHEMBL5206956)
Affinity DataKi:  470nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596982(CHEMBL5177471)
Affinity DataKi:  720nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596983(CHEMBL5190070)
Affinity DataKi:  730nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50568522(CHEMBL4864352)
Affinity DataKi:  750nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596974(CHEMBL5175317)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596972(CHEMBL5172654)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596975(CHEMBL5184132)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596976(CHEMBL5200476)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596977(CHEMBL5179061)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596985(CHEMBL5170156)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596978(CHEMBL5171912)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596979(CHEMBL5181710)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596984(CHEMBL5207485)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of MAO-A (unknown origin) using tyramine as substrate and measured after 10 mins by peroxidase-coupled reaction methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596985(CHEMBL5170156)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of MAO-A (unknown origin) using tyramine as substrate and measured after 10 mins by peroxidase-coupled reaction methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596984(CHEMBL5207485)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of MAO-B (unknown origin) using tyramine as substrate and measured after 10 mins by peroxidase-coupled reaction methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Riken Center For Sustainable Resource Science

Curated by ChEMBL
LigandPNGBDBM50596985(CHEMBL5170156)
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of MAO-B (unknown origin) using tyramine as substrate and measured after 10 mins by peroxidase-coupled reaction methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed