Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50016464
TargetPyruvate dehydrogenase complex component E2(Human)
National Cheng Kung University
Curated by ChEMBL
National Cheng Kung University
Curated by ChEMBL
Affinity DataKd: 578nMAssay Description:Binding affinity to recombinant GFP fused Dalt (unknown origin) by Lip-SMap analysisMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to recombinant human TrkB receptor ECD assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of porcine pancreatic lipase using trioleate as substrate assessed as inhibition of substrate hydrolysis measured for 10 minsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
National Cheng Kung University
Curated by ChEMBL
National Cheng Kung University
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
