Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50017779
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604970(CHEMBL5208940)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604970(CHEMBL5208940)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604983(CHEMBL5191108)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604983(CHEMBL5191108)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604982(CHEMBL5183680)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604982(CHEMBL5183680)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Rat)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604966(CHEMBL5175530)
Affinity DataKi:  5.10nMAssay Description:Binding affinity to rat sigma 2 receptor/TMEM97 expressed in rat PC-12 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604981(CHEMBL5197224)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604981(CHEMBL5197224)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604974(CHEMBL5206383)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604974(CHEMBL5206383)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604966(CHEMBL5175530)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604971(CHEMBL5177703)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604971(CHEMBL5177703)
Affinity DataKi:  8nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604966(CHEMBL5175530)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604979(CHEMBL5185602)
Affinity DataKi:  11nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604979(CHEMBL5185602)
Affinity DataKi:  11nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604970(CHEMBL5208940)
Affinity DataKi:  14nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604974(CHEMBL5206383)
Affinity DataKi:  14nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604970(CHEMBL5208940)
Affinity DataKi:  14nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604974(CHEMBL5206383)
Affinity DataKi:  15nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604976(CHEMBL5189334)
Affinity DataKi:  15nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604976(CHEMBL5189334)
Affinity DataKi:  16nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604972(CHEMBL5207336)
Affinity DataKi:  18nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604972(CHEMBL5207336)
Affinity DataKi:  18nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604979(CHEMBL5185602)
Affinity DataKi:  19nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604979(CHEMBL5185602)
Affinity DataKi:  19nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604971(CHEMBL5177703)
Affinity DataKi:  20nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604971(CHEMBL5177703)
Affinity DataKi:  20nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Rat)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604968(CHEMBL5190189)
Affinity DataKi:  23nMAssay Description:Binding affinity to rat sigma 2 receptor/TMEM97 expressed in rat PC-12 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604966(CHEMBL5175530)
Affinity DataKi:  29nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604966(CHEMBL5175530)
Affinity DataKi:  30nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604976(CHEMBL5189334)
Affinity DataKi:  32nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604976(CHEMBL5189334)
Affinity DataKi:  33nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604982(CHEMBL5183680)
Affinity DataKi:  38nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604982(CHEMBL5183680)
Affinity DataKi:  38nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Rat)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604969(CHEMBL5189158)
Affinity DataKi:  46nMAssay Description:Binding affinity to rat sigma 2 receptor/TMEM97 expressed in rat PC-12 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604975(CHEMBL5170591)
Affinity DataKi:  50nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604975(CHEMBL5170591)
Affinity DataKi:  50nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604972(CHEMBL5207336)
Affinity DataKi:  51nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604972(CHEMBL5207336)
Affinity DataKi:  52nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604983(CHEMBL5191108)
Affinity DataKi:  63nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604983(CHEMBL5191108)
Affinity DataKi:  63nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604981(CHEMBL5197224)
Affinity DataKi:  75nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604981(CHEMBL5197224)
Affinity DataKi:  76nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604975(CHEMBL5170591)
Affinity DataKi:  79nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604975(CHEMBL5170591)
Affinity DataKi:  79nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604973(CHEMBL5184025)
Affinity DataKi:  89nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604973(CHEMBL5184025)
Affinity DataKi:  90nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor/TMEM97 transfected in human HEK293T cells assessed as inhibition constant in pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Rat)
University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50604967(CHEMBL1698776)
Affinity DataKi:  90nMAssay Description:Binding affinity to rat sigma 2 receptor/TMEM97 expressed in rat PC-12 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
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