Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 50015398
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  200nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataKd:  150nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM439497(US10633379, Example 82 | US10633379, Example 35)
Affinity DataKd:  1.60nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM439497(US10633379, Example 82 | US10633379, Example 35)
Affinity DataKd:  520nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)
Affinity DataKd:  3.00E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) (N44 to E168 residues) expressed in bacterial expression system assessed as dissociation constant by BROMOsca...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)
Affinity DataKd:  63nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) (K333 to E460 residues) expressed in bacterial system assessed as dissociation constant by BROMOscan methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50: 20nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 2(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50: 71nMAssay Description:Inhibition of BRD2-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50543359(GSK620)
Affinity DataIC50: 72nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586230(CHEMBL5081350)
Affinity DataIC50: 72nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50: 85nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50544300(GSK046)
Affinity DataIC50: 98nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586228(CHEMBL5077541)
Affinity DataIC50: 100nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 2(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50: 120nMAssay Description:Inhibition of BRD2-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50: 130nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586226(CHEMBL5069987)
Affinity DataIC50: 140nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586236(CHEMBL5083228)
Affinity DataIC50: 150nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586243(CHEMBL5072385)
Affinity DataIC50: 170nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586242(CHEMBL5074953)
Affinity DataIC50: 170nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586239(CHEMBL5094390)
Affinity DataIC50: 210nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586238(CHEMBL5089658)
Affinity DataIC50: 210nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586233(CHEMBL5077199)
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586227(CHEMBL5079297)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586244(CHEMBL5086321)
Affinity DataIC50: 320nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50: 325nMAssay Description:Binding affinity to human partial length BRD3-BD2 (G306 to P416) expressed in bacterial system assessed as dissociation constant by BROMOscan methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586237(CHEMBL5075819)
Affinity DataIC50: 380nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586240(CHEMBL5076502)
Affinity DataIC50: 410nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586224(CHEMBL5085041)
Affinity DataIC50: 410nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586232(CHEMBL5089846)
Affinity DataIC50: 420nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586229(CHEMBL5089257)
Affinity DataIC50: 440nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586247(CHEMBL5075514)
Affinity DataIC50: 470nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586235(CHEMBL5094939)
Affinity DataIC50: 490nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586241(CHEMBL5090901)
Affinity DataIC50: 530nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586231(CHEMBL5090190)
Affinity DataIC50: 570nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586234(CHEMBL5081830)
Affinity DataIC50: 630nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586246(CHEMBL5074555)
Affinity DataIC50: 740nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50: 775nMAssay Description:Binding affinity to human partial length BRD4-BD2 (K333 to E460 residues) expressed in bacterial system assessed as dissociation constant by BROMOsca...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586219(CHEMBL5077591)
Affinity DataIC50: 800nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586245(CHEMBL5076250)
Affinity DataIC50: 880nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50: 900nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586216(CHEMBL5078986)
Affinity DataIC50: 900nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586220(CHEMBL5084945)
Affinity DataIC50: 900nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586221(CHEMBL5075052)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586217(CHEMBL5084236)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586222(CHEMBL5082786)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586245(CHEMBL5076250)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586218(CHEMBL5093626)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586244(CHEMBL5086321)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586231(CHEMBL5090190)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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