Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50017673
TargetBeta-2 adrenergic receptor(Human)
Northwest University

Curated by ChEMBL
LigandPNGBDBM50603973(CHEMBL5172549)
Affinity DataKd:  7.5nMAssay Description:Binding affinity to immobilized Halo tag-fused beta2 adrenoceptor (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBeta-2 adrenergic receptor(Human)
Northwest University

Curated by ChEMBL
LigandPNGBDBM50595336(Methoxyphenamine | METHOXYPHENAMINE)
Affinity DataKd:  0.980nMAssay Description:Binding affinity to immobilized Halo tag-fused beta2 adrenoceptor (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
Northwest University

Curated by ChEMBL
LigandPNGBDBM50603973(CHEMBL5172549)
Affinity DataKd:  17nMAssay Description:Binding affinity to immobilized Halo tag-fused CysLT receptor (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation rate...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
Northwest University

Curated by ChEMBL
LigandPNGBDBM50239015(CHEBI:6993 | MK-476 | Montelukast Sodium | Singula...)
Affinity DataKd:  13nMAssay Description:Binding affinity to immobilized Halo tag-fused CysLT receptor (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation rate...More data for this Ligand-Target Pair
In DepthDetails
PubMed