Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50017664
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataEC50:  2.92E+3nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 6-OAU-induced calcium response curve b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataEC50:  2.84E+4nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 3-OH-C12-induced calcium response curv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataEC50:  2.21E+4nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 3-OH-C12-induced calcium response curv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataEC50:  8.42E+4nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 3-OH-C12-induced calcium response curv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataEC50:  4.86E+4nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 3-OH-C12-induced calcium response curv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataEC50:  4.87E+5nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 3-OH-C12-induced calcium response curv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataEC50:  9.24E+4nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 3-OH-C12-induced calcium response curv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataEC50:  1.13E+3nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 6-OAU-induced calcium response curve b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataEC50:  611nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 6-OAU-induced calcium response curve b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataEC50:  1.79E+3nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 6-OAU-induced calcium response curve b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataEC50:  655nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 6-OAU-induced calcium response curve b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataEC50:  3.73E+3nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as right shift in 6-OAU-induced calcium response curve b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603899(CHEMBL5205352)
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603880(CHEMBL5191944)
Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603901(CHEMBL5176994)
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603875(CHEMBL5206571)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603904(CHEMBL5197375)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603900(CHEMBL5190809)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603881(CHEMBL5202207)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603891(CHEMBL5170437)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603902(CHEMBL5201979)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603868(CHEMBL5201755)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603882(CHEMBL5171959)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603886(CHEMBL5192281)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603892(CHEMBL5195150)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603877(CHEMBL5183789)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603883(CHEMBL5198754)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603903(CHEMBL5175363)
Affinity DataIC50: 56nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataIC50: 58nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells assessed as reversal of 6-OAU induced inhibition of forskolin induced intracellular cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603887(CHEMBL5192624)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603869(CHEMBL5194984)
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603896(CHEMBL5187339)
Affinity DataIC50: 89nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603885(CHEMBL5177531)
Affinity DataIC50: 89nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataIC50: 107nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells assessed as reversal of 6-OAU induced inhibition of forskolin induced intracellular cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50548385(Glpg-1205 | Glpg1205)
Affinity DataIC50: 112nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603897(CHEMBL5196560)
Affinity DataIC50: 114nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603869(CHEMBL5194984)
Affinity DataIC50: 118nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 3-OH-C12 induced intracellular calcium r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603873(CHEMBL5189167)
Affinity DataIC50: 146nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603890(CHEMBL5203023)
Affinity DataIC50: 165nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603878(CHEMBL5179740)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603889(CHEMBL5190004)
Affinity DataIC50: 234nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50556781(CHEMBL3719364)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human GPR84 expressed in CHO-K1 cells assessed as reduction in 6-OAU induced intracellular cAMP production pretreated for 15 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603879(CHEMBL5170786)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Mouse)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603895(CHEMBL5179395)
Affinity DataIC50: 273nMAssay Description:Antagonist activity at mouse GPR84 expressed in HEK293 cells assessed as reduction in 6-OAU induced intracellular calcium response preincubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603894(CHEMBL5184044)
Affinity DataIC50: 277nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603893(CHEMBL5198261)
Affinity DataIC50: 305nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603884(CHEMBL5195223)
Affinity DataIC50: 321nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603888(CHEMBL5207051)
Affinity DataIC50: 328nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetG-protein coupled receptor 84(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50603906(CHEMBL5170482)
Affinity DataIC50: 345nMAssay Description:Antagonist activity at human GPR84 expressed in HEK293 cells co-expressing Galpha16 assessed as reduction in 6-OAU induced intracellular calcium resp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
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